Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
ADORA1 134 TECADENOSON CHEMBL392149 agonist TdgClinicalTrial, ChemblInteractions, DrugBank, TTD 16230891, 13678937, 15956124
ADORA1 134 CAFFEINE, CITRATED CHEMBL1200569 antagonist ChemblInteractions
ADORA1 134 AMINOPHYLLINE CHEMBL1370561 antagonist ChemblInteractions, DrugBank 12735630, 8425287
ADORA1 134 GW493838 CHEMBL3545223 agonist ChemblInteractions
ADORA1 134 ADENOSINE CHEMBL477 agonist GuideToPharmacologyInteractions, ChemblInteractions
ADORA1 134 THEOPHYLLINE SODIUM GLYCINATE CHEMBL1200578 antagonist ChemblInteractions
ADORA1 134 Derenofylline CHEMBL592435 antagonist GuideToPharmacologyInteractions, ChemblInteractions, TTD
ADORA1 134 GS-9667 CHEMBL3545011 partial agonist TdgClinicalTrial, ChemblInteractions
ADORA1 134 AMP579 CHEMBL3545163 agonist ChemblInteractions
ADORA1 134 CHEMBL257833 CHEMBL257833 agonist GuideToPharmacologyInteractions
ADORA1 134 REGADENOSON CHEMBL317052 agonist GuideToPharmacologyInteractions
ADORA1 134 N6-CYCLOPENTYLADENOSINE CHEMBL68738 agonist GuideToPharmacologyInteractions
ADORA1 134 CGS-21680 CHEMBL331372 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL59532 CHEMBL59532 allosteric modulator GuideToPharmacologyInteractions
ADORA1 134 CGS-15943 CHEMBL16687 antagonist GuideToPharmacologyInteractions
ADORA1 134 ISTRADEFYLLINE CHEMBL431770 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL375293 CHEMBL375293 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL219160 CHEMBL219160 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL273807 CHEMBL273807 antagonist GuideToPharmacologyInteractions
ADORA1 134 IMISOPASEM MANGANESE CHEMBL3544979 antagonist GuideToPharmacologyInteractions
ADORA1 134 VIPADENANT CHEMBL447664 antagonist GuideToPharmacologyInteractions
ADORA1 134 ZM-241385 CHEMBL113142 antagonist GuideToPharmacologyInteractions
ADORA1 134 THEOBROMINE CHEMBL1114 antagonist DrugBank 16702031, 12602592, 17085856, 17372967, 17126319, 17162470, 15095008, 3588607
ADORA1 134 DEFIBROTIDE CHEMBL2108396 DrugBank 8405101
ADORA1 134 CHEMBL57997 CHEMBL57997 TdgClinicalTrial
ADORA1 134 RPR749 CHEMBL3545331 agonist ChemblInteractions
ADORA1 134 BINODENOSON CHEMBL1950554 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL1895774 CHEMBL1895774 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL175788 CHEMBL175788 agonist GuideToPharmacologyInteractions
ADORA1 134 8-CYCLOPENTYLTHEOPHYLLINE CHEMBL106265 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL2311146 CHEMBL2311146 antagonist GuideToPharmacologyInteractions
ADORA1 134 GS 6201 CHEMBL260933 antagonist GuideToPharmacologyInteractions
ADORA1 134 1,3-DIPROPYL-8-CYCLOPENTYLXANTHINE [DPCPX] CHEMBL183 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL111545 CHEMBL111545 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL1562432 CHEMBL1562432 antagonist GuideToPharmacologyInteractions
ADORA1 134 XANTHINE AMINE CONGENER CHEMBL273094 antagonist GuideToPharmacologyInteractions
ADORA1 134 DYPHYLLINE CHEMBL1752 antagonist DrugBank 2997628
ADORA1 134 GABAPENTIN CHEMBL940 agonist DrugBank 15765150, 15140630, 15572277
ADORA1 134 ROLOFYLLINE (CHEMBL2103819) CHEMBL2103819 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
ADORA1 134 TONAPOFYLLINE CHEMBL414157 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
ADORA1 134 Trabodenoson CHEMBL3545407 agonist TdgClinicalTrial, ChemblInteractions
ADORA1 134 APADENOSON CHEMBL1950649 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL260563 CHEMBL260563 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL285819 CHEMBL285819 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL410873 CHEMBL410873 agonist GuideToPharmacologyInteractions
ADORA1 134 NECA CHEMBL464859 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL302765 CHEMBL302765 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL8565 CHEMBL8565 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL136689 CHEMBL136689 antagonist GuideToPharmacologyInteractions
ADORA1 134 PBF-680 CHEMBL3545162 antagonist ChemblInteractions
ADORA1 134 NAXIFYLLINE CHEMBL2107805 antagonist ChemblInteractions, DrugBank, TTD
ADORA1 134 ROLOFYLLINE (CHEMBL52333) CHEMBL52333 antagonist TTD
ADORA1 134 FK453 CHEMBL440115 antagonist GuideToPharmacologyInteractions, ChemblInteractions
ADORA1 134 SELODENOSON CHEMBL2107371 agonist ChemblInteractions
ADORA1 134 BAY1067197 CHEMBL3545405 agonist ChemblInteractions
ADORA1 134 CAFFEINE CHEMBL113 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, TTD
ADORA1 134 Capadenoson CHEMBL3235279 partial agonist ChemblInteractions
ADORA1 134 CF102 CHEMBL431733 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL175543 CHEMBL175543 agonist GuideToPharmacologyInteractions
ADORA1 134 (R)-PIA CHEMBL139000 agonist GuideToPharmacologyInteractions
ADORA1 134 (S)-PIA CHEMBL420705 agonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL284969 CHEMBL284969 agonist GuideToPharmacologyInteractions
ADORA1 134 ISOBUTYLMETHYLXANTHINE CHEMBL275084 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL2181965 CHEMBL2181965 antagonist GuideToPharmacologyInteractions
ADORA1 134 CHEMBL89852 CHEMBL89852 antagonist GuideToPharmacologyInteractions
ADORA1 134 PRELADENANT CHEMBL240624 antagonist GuideToPharmacologyInteractions
ADORA1 134 ST1535 CHEMBL197669 antagonist GuideToPharmacologyInteractions
ADORA1 134 PENTOXIFYLLINE CHEMBL628 antagonist TdgClinicalTrial, DrugBank 3588607
ADORA1 134 THEOPHYLLINE CHEMBL190 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank 14992338, 3588607
ADORA1 134 ENPROFYLLINE CHEMBL279898 DrugBank 10496952
ADORA1 134 OXTRIPHYLLINE CHEMBL1200434 antagonist ChemblInteractions, DrugBank 14992338, 3588607

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID