Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
ADRA1B 147 METHOXAMINE CHEMBL524 agonist, stimulator TdgClinicalTrial, GuideToPharmacologyInteractions, TEND, DrugBank, TTD 11752352, 2546049, 11331292, 8635240, 2988814
ADRA1B 147 PROPIOMAZINE CHEMBL1201210 antagonist TdgClinicalTrial, TEND, DrugBank 17139284, 17016423
ADRA1B 147 DOXAZOSIN CHEMBL707 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND
ADRA1B 147 XYLOMETAZOLINE CHEMBL312448 agonist DrugBank 20030735
ADRA1B 147 LISDEXAMFETAMINE CHEMBL1201222 antagonist TdgClinicalTrial, TEND, TTD
ADRA1B 147 LABETALOL HYDROCHLORIDE CHEMBL1200323 antagonist ChemblInteractions
ADRA1B 147 EPINEPHRINE CHEMBL679 agonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
ADRA1B 147 ERGOLOID MESYLATES CHEMBL2311030 antagonist ChemblInteractions
ADRA1B 147 TETRAHYDROZOLINE HYDROCHLORIDE CHEMBL1200413 agonist ChemblInteractions
ADRA1B 147 PRAZOSIN CHEMBL2 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND
ADRA1B 147 BETHANIDINE CHEMBL1201260 TdgClinicalTrial, TEND
ADRA1B 147 TAMSULOSIN CHEMBL836 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND
ADRA1B 147 QUETIAPINE CHEMBL716 TEND
ADRA1B 147 MIDODRINE HYDROCHLORIDE CHEMBL1200461 agonist ChemblInteractions
ADRA1B 147 DOXAZOSIN MESYLATE CHEMBL1200561 antagonist ChemblInteractions
ADRA1B 147 CARVEDILOL PHOSPHATE CHEMBL1201167 antagonist ChemblInteractions
ADRA1B 147 LISDEXAMFETAMINE DIMESYLATE CHEMBL1201178 TdgClinicalTrial
ADRA1B 147 PHENYLEPHRINE BITARTRATE CHEMBL2062264 agonist ChemblInteractions
ADRA1B 147 ALFUZOSIN HYDROCHLORIDE CHEMBL1723 agonist ChemblInteractions
ADRA1B 147 CYPROHEPTADINE CHEMBL516 antagonist GuideToPharmacologyInteractions
ADRA1B 147 MIANSERIN CHEMBL6437 antagonist GuideToPharmacologyInteractions
ADRA1B 147 CHEMBL24777 CHEMBL24777 antagonist GuideToPharmacologyInteractions
ADRA1B 147 (+)-CYCLAZOSIN CHEMBL2261604 antagonist GuideToPharmacologyInteractions
ADRA1B 147 SPIPERONE CHEMBL267930 antagonist GuideToPharmacologyInteractions
ADRA1B 147 NOREPINEPHRINE CHEMBL1437 agonist TdgClinicalTrial, TEND, DrugBank 17139284, 17016423, 17266602, 18064417, 8166240, 8294418, 7773533
ADRA1B 147 CLOZAPINE CHEMBL42 antagonist GuideToPharmacologyInteractions, DrugBank 17848919
ADRA1B 147 PROMAZINE CHEMBL564 antagonist TdgClinicalTrial, TEND, DrugBank 17139284, 17016423
ADRA1B 147 LEVOMEPROMAZINE CHEMBL1764 antagonist TdgClinicalTrial, TEND, DrugBank 2870716, 15701205
ADRA1B 147 PERICIAZINE CHEMBL251940 antagonist, binder TdgClinicalTrial, TEND, DrugBank, TTD 11752352, 17139284, 17016423
ADRA1B 147 BREXPIPRAZOLE CHEMBL2105760 antagonist DrugBank 25225185
ADRA1B 147 MEPHENTERMINE SULFATE CHEMBL1200996 agonist ChemblInteractions
ADRA1B 147 NAPHAZOLINE HYDROCHLORIDE CHEMBL1706 agonist ChemblInteractions
ADRA1B 147 PHENOXYBENZAMINE HYDROCHLORIDE CHEMBL1200787 antagonist ChemblInteractions
ADRA1B 147 SENREBOTASE CHEMBL3137348 TdgClinicalTrial
ADRA1B 147 DEXTROAMPHETAMINE CHEMBL612 antagonist TTD
ADRA1B 147 LABETALOL CHEMBL429 TdgClinicalTrial, TEND
ADRA1B 147 NEFAZODONE CHEMBL623 TdgClinicalTrial, TEND
ADRA1B 147 PHENTOLAMINE MESYLATE CHEMBL1200873 antagonist ChemblInteractions
ADRA1B 147 ALFUZOSIN CHEMBL709 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND
ADRA1B 147 RAUWOLFIA SERPENTINA (CHEMBL3559672) CHEMBL3559672 antagonist ChemblInteractions
ADRA1B 147 TRIMIPRAMINE MALEATE CHEMBL1200948 antagonist ChemblInteractions
ADRA1B 147 OXYMETAZOLINE CHEMBL762 agonist GuideToPharmacologyInteractions
ADRA1B 147 NS-49 CHEMBL72958 agonist GuideToPharmacologyInteractions
ADRA1B 147 A-119637 CHEMBL268758 antagonist GuideToPharmacologyInteractions
ADRA1B 147 KETANSERIN CHEMBL51 antagonist GuideToPharmacologyInteractions
ADRA1B 147 UPIDOSIN CHEMBL278865 antagonist GuideToPharmacologyInteractions
ADRA1B 147 OXYMETAZOLINE HYDROCHLORIDE CHEMBL1200791 agonist ChemblInteractions
ADRA1B 147 ARIPIPRAZOLE CHEMBL1112 antagonist DrugBank 17848919
ADRA1B 147 RISPERIDONE CHEMBL85 antagonist GuideToPharmacologyInteractions, DrugBank 7691623, 11132243, 11752352, 15907153, 15992090, 8925876
ADRA1B 147 MODAFINIL CHEMBL1373 partial agonist DrugBank 17681557
ADRA1B 147 ACEPROMAZINE CHEMBL39560 antagonist DrugBank 15695070
ADRA1B 147 DRONEDARONE CHEMBL184412 antagonist DrugBank 17389667
ADRA1B 147 ALBIFLORIN CHEMBL1939883 DrugBank
ADRA1B 147 CHEMBL609728 CHEMBL609728 DrugBank
ADRA1B 147 DROXIDOPA CHEMBL2103827 agonist ChemblInteractions, DrugBank 8166240, 17266602, 20412040, 7773533
ADRA1B 147 HYDROXYAMPHETAMINE HYDROBROMIDE CHEMBL1200705 agonist ChemblInteractions
ADRA1B 147 MIDODRINE CHEMBL1201212 TdgClinicalTrial, TEND
ADRA1B 147 PHENDIMETRAZINE CHEMBL1744 antagonist TdgClinicalTrial, TEND, TTD
ADRA1B 147 TERAZOSIN HYDROCHLORIDE HYDRATE CHEMBL1201091 antagonist ChemblInteractions
ADRA1B 147 ERGOTAMINE TARTRATE CHEMBL2062265 agonist ChemblInteractions
ADRA1B 147 PHENYLEPHRINE HYDROCHLORIDE CHEMBL1200339 agonist ChemblInteractions
ADRA1B 147 CHEMBL420060 CHEMBL420060 antagonist GuideToPharmacologyInteractions
ADRA1B 147 INDORAMIN CHEMBL279516 antagonist GuideToPharmacologyInteractions
ADRA1B 147 L-765314 CHEMBL19476 antagonist GuideToPharmacologyInteractions
ADRA1B 147 CHEMBL1256701 CHEMBL1256701 antagonist GuideToPharmacologyInteractions
ADRA1B 147 RITANSERIN CHEMBL267777 antagonist GuideToPharmacologyInteractions
ADRA1B 147 NIGULDIPINE CHEMBL405355 antagonist GuideToPharmacologyInteractions
ADRA1B 147 ALSEROXYLON CHEMBL1201454 antagonist ChemblInteractions
ADRA1B 147 TOLAZOLINE HYDROCHLORIDE CHEMBL1689 antagonist ChemblInteractions
ADRA1B 147 METARAMINOL BITARTRATE CHEMBL2062262 agonist ChemblInteractions
ADRA1B 147 DAPIPRAZOLE CHEMBL1201216 antagonist TdgClinicalTrial, TEND, DrugBank 17139284, 17016423
ADRA1B 147 OLANZAPINE CHEMBL715 antagonist TdgClinicalTrial, TEND, DrugBank 11752352, 17316700, 17848919, 10227113
ADRA1B 147 LOXAPINE CHEMBL831 binder DrugBank
ADRA1B 147 FENOLDOPAM CHEMBL588 DrugBank 7670737
ADRA1B 147 CARVEDILOL CHEMBL723 antagonist ChemblInteractions, DrugBank 15306222
ADRA1B 147 PALIPERIDONE CHEMBL1621 antagonist DrugBank 7691623, 11132243, 15907153, 7531353, 7524043, 15992090, 8925876, 18542932
ADRA1B 147 THIOPROPERAZINE CHEMBL609109 antagonist DrugBank 15695070
ADRA1B 147 CIRAZOLINE CHEMBL13852 partial agonist DrugBank 8564227, 6123592
ADRA1B 147 NORADRENALINE CHEMBL1356607 agonist ChemblInteractions
ADRA1B 147 PHENYLEPHRINE CHEMBL1215 agonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND
ADRA1B 147 TERAZOSIN CHEMBL611 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND
ADRA1B 147 DEBRISOQUIN CHEMBL169901 TdgClinicalTrial, TEND
ADRA1B 147 METHAMPHETAMINE CHEMBL1201201 antagonist TEND, TTD
ADRA1B 147 TRAZODONE CHEMBL621 TEND
ADRA1B 147 TAMSULOSIN HYDROCHLORIDE CHEMBL1200914 antagonist ChemblInteractions
ADRA1B 147 EPINEPHRINE BITARTRATE CHEMBL1256958 agonist ChemblInteractions
ADRA1B 147 DIPIVEFRIN HYDROCHLORIDE CHEMBL1200833 agonist ChemblInteractions
ADRA1B 147 PRAZOSIN HYDROCHLORIDE CHEMBL1558 antagonist ChemblInteractions
ADRA1B 147 METHOXAMINE HYDROCHLORIDE CHEMBL1201103 agonist ChemblInteractions
ADRA1B 147 A-123189 CHEMBL13856 antagonist GuideToPharmacologyInteractions
ADRA1B 147 BMY-7378 CHEMBL13647 antagonist GuideToPharmacologyInteractions
ADRA1B 147 PHENTOLAMINE CHEMBL597 antagonist GuideToPharmacologyInteractions
ADRA1B 147 SPIROXATRINE CHEMBL300555 antagonist GuideToPharmacologyInteractions
ADRA1B 147 CHEMBL25554 CHEMBL25554 antagonist GuideToPharmacologyInteractions
ADRA1B 147 ERGOTAMINE CHEMBL442 partial agonist DrugBank 18066532
ADRA1B 147 SILODOSIN CHEMBL24778 antagonist GuideToPharmacologyInteractions, DrugBank 21114397
ADRA1B 147 SERTINDOLE CHEMBL12713 TdgClinicalTrial, TEND, DrugBank 16925508
ADRA1B 147 CABERGOLINE CHEMBL1201087 binder DrugBank 12388666

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID