Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GRIA2 2891 BUTABARBITAL CHEMBL449 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 SECOBARBITAL CHEMBL447 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 THIOPENTAL CHEMBL441 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 PRIMIDONE CHEMBL856 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 PHENOBARBITAL CHEMBL40 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449, 20051697
GRIA2 2891 CHEMBL1255648 CHEMBL1255648 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 CYCLOTHIAZIDE CHEMBL61593 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 CHEMBL320642 CHEMBL320642 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 BECAMPANEL CHEMBL2107735 antagonist ChemblInteractions
GRIA2 2891 PENTOBARBITAL CHEMBL448 TdgClinicalTrial, TEND
GRIA2 2891 MIBAMPATOR CHEMBL1277001 positive allosteric modulator ChemblInteractions
GRIA2 2891 BUTALBITAL CHEMBL454 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 CHEMBL136800 CHEMBL136800 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 CHEMBL77862 CHEMBL77862 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 CHEMBL1097939 CHEMBL1097939 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 PIRACETAM CHEMBL36715 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 NBQX CHEMBL222519 antagonist GuideToPharmacologyInteractions
GRIA2 2891 AMOBARBITAL CHEMBL267894 antagonist DrugBank 10487207, 11264449
GRIA2 2891 APROBARBITAL CHEMBL7863 antagonist DrugBank 10487207, 11264449
GRIA2 2891 HEPTABARBITAL CHEMBL468837 antagonist DrugBank 10487207, 11264449
GRIA2 2891 CHEMBL594840 CHEMBL594840 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 QUISQUALATE CHEMBL279956 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 CHEMBL27130 CHEMBL27130 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 DNQX CHEMBL155265 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 IRAMPANEL CHEMBL29741 antagonist ChemblInteractions
GRIA2 2891 MK-8777 CHEMBL3707401 positive allosteric modulator ChemblInteractions
GRIA2 2891 PF-04958242 CHEMBL3707379 positive allosteric modulator ChemblInteractions
GRIA2 2891 Selurampanel CHEMBL3545042 antagonist TdgClinicalTrial, ChemblInteractions
GRIA2 2891 BUTETHAL CHEMBL404422 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 L-GLUTAMATE CHEMBL575060 DrugBank 17139284, 17016423, 1279377, 7838123, 7679210
GRIA2 2891 TALBUTAL CHEMBL1200802 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 MEPHOBARBITAL CHEMBL45029 antagonist DrugBank 10487207, 11264449
GRIA2 2891 ANIRACETAM CHEMBL36994 allosteric modulator GuideToPharmacologyInteractions, DrugBank 10592235
GRIA2 2891 CHEMBL222418 CHEMBL222418 antagonist GuideToPharmacologyInteractions
GRIA2 2891 BARBITAL CHEMBL444 antagonist DrugBank 10487207, 11264449
GRIA2 2891 CHEMBL121915 CHEMBL121915 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 CHEMBL333964 CHEMBL333964 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 (S)-WILLARDIINE CHEMBL122005 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 CHEMBL28472 CHEMBL28472 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 CX1739 CHEMBL3707399 positive allosteric modulator ChemblInteractions
GRIA2 2891 DASOLAMPANEL CHEMBL2103869 antagonist ChemblInteractions
GRIA2 2891 FARAMPATOR CHEMBL1276138 positive allosteric modulator ChemblInteractions
GRIA2 2891 METHARBITAL CHEMBL450 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 (R,S)-AMPA CHEMBL13378 agonist GuideToPharmacologyInteractions
GRIA2 2891 CHEMBL123132 CHEMBL123132 agonist GuideToPharmacologyInteractions, DrugBank 17139284, 17016423, 10592235
GRIA2 2891 CHEMBL334920 CHEMBL334920 allosteric modulator GuideToPharmacologyInteractions
GRIA2 2891 CHEMBL265301 CHEMBL265301 antagonist GuideToPharmacologyInteractions
GRIA2 2891 GYKI-52466 CHEMBL275006 antagonist GuideToPharmacologyInteractions
GRIA2 2891 TEZAMPANEL CHEMBL14935 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions
GRIA2 2891 HEXOBARBITAL CHEMBL7728 antagonist TdgClinicalTrial, TEND, DrugBank 10487207, 11264449
GRIA2 2891 (S)-AMPA CHEMBL276815 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 CHEMBL337577 CHEMBL337577 DrugBank 17139284, 17016423, 10592235
GRIA2 2891 PERAMPANEL CHEMBL1214124 antagonist TdgClinicalTrial, ChemblInteractions
GRIA2 2891 ZONAMPANEL CHEMBL119625 antagonist ChemblInteractions
GRIA2 2891 TOPIRAMATE CHEMBL220492 antagonist ChemblInteractions
GRIA2 2891 TALAMPANEL CHEMBL61872 TdgClinicalTrial, DrugBank 12581229, 17199027, 16861112

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID