Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
HRH2 3274 CIMETIDINE CHEMBL30 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, TTD
HRH2 3274 NIZATIDINE CHEMBL653 antagonist TdgClinicalTrial, ChemblInteractions, TEND, DrugBank, TTD 1843561, 2895808, 11752352, 2877081, 2858133, 2567267
HRH2 3274 ARPROMIDINE CHEMBL293802 agonist GuideToPharmacologyInteractions
HRH2 3274 TIPROLISANT CHEMBL462605 antagonist GuideToPharmacologyInteractions
HRH2 3274 CHEMBL351231 CHEMBL351231 antagonist GuideToPharmacologyInteractions
HRH2 3274 TOLAZOLINE HYDROCHLORIDE CHEMBL1689 agonist ChemblInteractions
HRH2 3274 BETAZOLE HYDROCHLORIDE CHEMBL1200949 agonist ChemblInteractions
HRH2 3274 BETAZOLE CHEMBL1201323 agonist, antagonist TdgClinicalTrial, TEND, DrugBank, TTD 2892392, 2886642, 11752352, 7213132, 2874214, 3661710
HRH2 3274 LOXAPINE CHEMBL831 binder DrugBank
HRH2 3274 METHANTHELINE CHEMBL1201264 antagonist DrugBank 6116801
HRH2 3274 CLOBENPROPIT CHEMBL14690 antagonist GuideToPharmacologyInteractions
HRH2 3274 MK-0249 CHEMBL476323 antagonist GuideToPharmacologyInteractions
HRH2 3274 DOXEPIN CHEMBL1628227 TdgClinicalTrial
HRH2 3274 EPINASTINE CHEMBL1106 TdgClinicalTrial, TEND
HRH2 3274 FAMOTIDINE CHEMBL902 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank, TTD 16513821, 12509588, 16702624, 16723495, 11752352, 1646056, 18310651, 2067140, 19578661, 12832840, 17273750
HRH2 3274 CIMETIDINE HYDROCHLORIDE CHEMBL1201051 antagonist ChemblInteractions
HRH2 3274 HISTAMINE CHEMBL90 agonist TdgClinicalTrial, DrugBank 17334413, 11752352, 17359382
HRH2 3274 BURIMAMIDE CHEMBL12160 agonist GuideToPharmacologyInteractions
HRH2 3274 CHEMBL472273 CHEMBL472273 agonist GuideToPharmacologyInteractions
HRH2 3274 ASENAPINE (CHEMBL3187365) CHEMBL3187365 TdgClinicalTrial
HRH2 3274 METHANTHELINE BROMIDE CHEMBL1200988 antagonist ChemblInteractions
HRH2 3274 RANITIDINE HYDROCHLORIDE CHEMBL2110372 antagonist ChemblInteractions
HRH2 3274 TOLAZOLINE CHEMBL770 agonist DrugBank 21948594, 8487790, 6386273
HRH2 3274 ROXATIDINE ACETATE CHEMBL46102 antagonist DrugBank 20718616
HRH2 3274 AMTHAMINE CHEMBL293762 agonist GuideToPharmacologyInteractions
HRH2 3274 IMPROMIDINE CHEMBL12608 agonist GuideToPharmacologyInteractions
HRH2 3274 CHEMBL513056 CHEMBL513056 agonist GuideToPharmacologyInteractions
HRH2 3274 CIPROXIFAN CHEMBL14638 antagonist GuideToPharmacologyInteractions
HRH2 3274 CONESSINE CHEMBL191703 antagonist GuideToPharmacologyInteractions
HRH2 3274 NAFCILLIN CHEMBL1443 antagonist GuideToPharmacologyInteractions
HRH2 3274 RANITIDINE CHEMBL1790041 antagonist TdgClinicalTrial, GuideToPharmacologyInteractions, TEND, TTD
HRH2 3274 TIOTIDINE CHEMBL269646 antagonist GuideToPharmacologyInteractions
HRH2 3274 RANITIDINE BISMUTH CITRATE CHEMBL2111286 antagonist ChemblInteractions
HRH2 3274 OLANZAPINE CHEMBL715 antagonist DrugBank 18308814
HRH2 3274 METIAMIDE CHEMBL275446 antagonist DrugBank 7725982

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID