Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
PDE4A 5141 CRISABOROLE CHEMBL484785 inhibitor TdgClinicalTrial, ChemblInteractions, DrugBank
PDE4A 5141 CHEMBL74078 CHEMBL74078 DrugBank 10592235
PDE4A 5141 CDP840 CHEMBL32442 inhibitor GuideToPharmacologyInteractions
PDE4A 5141 ENPROFYLLINE CHEMBL279898 inhibitor TdgClinicalTrial, TEND, DrugBank, TTD 2262902, 1885257, 11752352, 3446047, 17670210, 3002801
PDE4A 5141 SODIUM PHENYLBUTYRATE CHEMBL1746 inhibitor GuideToPharmacologyInteractions
PDE4A 5141 CHEMBL1232082 CHEMBL1232082 inhibitor GuideToPharmacologyInteractions
PDE4A 5141 MILRINONE CHEMBL189 TdgClinicalTrial, TEND
PDE4A 5141 CHEMBL570015 CHEMBL570015 inhibitor TTD
PDE4A 5141 PERAMIVIR CHEMBL139367 inhibitor TTD
PDE4A 5141 THEOPHYLLINE CHEMBL190 inhibitor TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 12887610, 15351234, 12421478, 12547256, 15253881
PDE4A 5141 IBUDILAST CHEMBL19449 inhibitor TdgClinicalTrial, GuideToPharmacologyInteractions, DrugBank 21036126, 16313925, 20124930
PDE4A 5141 CHEMBL1229585 CHEMBL1229585 DrugBank 10592235
PDE4A 5141 CHEMBL1358525 CHEMBL1358525 inhibitor GuideToPharmacologyInteractions
PDE4A 5141 THEOPHYLLINE SODIUM GLYCINATE CHEMBL1200578 inhibitor ChemblInteractions
PDE4A 5141 AMINOPHYLLINE CHEMBL1370561 inhibitor ChemblInteractions
PDE4A 5141 CILOMILAST CHEMBL511115 inhibitor TTD
PDE4A 5141 FLAVOXATE HYDROCHLORIDE CHEMBL1200875 inhibitor ChemblInteractions
PDE4A 5141 SAFRAMYCIN A CHEMBL452709 inhibitor TTD
PDE4A 5141 AROFYLLINE CHEMBL1598450 inhibitor TTD
PDE4A 5141 ETAZOLATE CHEMBL356388 TdgClinicalTrial
PDE4A 5141 PENTOXIFYLLINE CHEMBL628 inhibitor TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 11752352
PDE4A 5141 DYPHYLLINE CHEMBL1752 inhibitor TdgClinicalTrial, ChemblInteractions, TEND, DrugBank, TTD 7925603, 11752352, 17139284, 17016423, 225216
PDE4A 5141 DIPYRIDAMOLE CHEMBL932 inhibitor TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 11752352
PDE4A 5141 OXTRIPHYLLINE CHEMBL1200434 inhibitor ChemblInteractions, DrugBank 12887610, 15351234, 12421478, 12547256, 15253881
PDE4A 5141 DROTAVERINE CHEMBL551978 inhibitor DrugBank 12823389, 17502703, 20554370
PDE4A 5141 ROLIPRAM CHEMBL63 inhibitor GuideToPharmacologyInteractions
PDE4A 5141 TADALAFIL CHEMBL779 TEND
PDE4A 5141 AMLEXANOX CHEMBL1096 inhibitor ChemblInteractions
PDE4A 5141 ILOPROST CHEMBL494 inducer DrugBank 2461561, 12441759, 11551870, 12952271
PDE4A 5141 ROFLUMILAST CHEMBL193240 inhibitor TdgClinicalTrial, ChemblInteractions, DrugBank, TTD 17726343
PDE4A 5141 PICLAMILAST CHEMBL42126 DrugBank 15765929
PDE4A 5141 APREMILAST CHEMBL514800 antagonist, inhibitor TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, DrugBank, TTD 25864487, 17352685
PDE4A 5141 TOFISOPAM CHEMBL404216 inhibitor DrugBank 20967473

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID