Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
PIK3R2 5296 PA-799 CHEMBL1684984 inhibitor ChemblInteractions
PIK3R2 5296 COPANLISIB CHEMBL3218576 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R2 5296 OMIPALISIB CHEMBL1236962 inhibitor MyCancerGenomeClinicalTrial, ChemblInteractions
PIK3R2 5296 RECILISIB CHEMBL2219421 inhibitor ChemblInteractions
PIK3R2 5296 Panulisib CHEMBL3545322 inhibitor ChemblInteractions
PIK3R2 5296 ZSTK-474 CHEMBL586701 inhibitor ChemblInteractions
PIK3R2 5296 PICTILISIB CHEMBL521851 inhibitor MyCancerGenome, ChemblInteractions
PIK3R2 5296 BUPARLISIB CHEMBL2017974 inhibitor MyCancerGenome, ChemblInteractions
PIK3R2 5296 WX-037 CHEMBL3545385 inhibitor ChemblInteractions
PIK3R2 5296 ISOPRENALINE CHEMBL1160723 agonist DrugBank 15110780, 15618457, 15381832, 15527548, 15985706
PIK3R2 5296 PWT-33587 CHEMBL3545006 inhibitor ChemblInteractions
PIK3R2 5296 VOXTALISIB CHEMBL3545366 inhibitor MyCancerGenome, ChemblInteractions
PIK3R2 5296 GSK-2636771 CHEMBL3188551 inhibitor MyCancerGenome
PIK3R2 5296 PILARALISIB (CHEMBL3218575) CHEMBL3218575 inhibitor MyCancerGenome
PIK3R2 5296 LY-3023414 CHEMBL3544999 inhibitor ChemblInteractions
PIK3R2 5296 BUPARLISIB HYDROCHLORIDE CHEMBL2364604 inhibitor MyCancerGenomeClinicalTrial
PIK3R2 5296 RG-7666 CHEMBL3545324 inhibitor ChemblInteractions
PIK3R2 5296 PF-04691502 CHEMBL1234354 inhibitor MyCancerGenome, ChemblInteractions
PIK3R2 5296 SF-1126 CHEMBL2326966 inhibitor MyCancerGenome, ChemblInteractions, DrugBank
PIK3R2 5296 DS-7423 CHEMBL3545248 inhibitor ChemblInteractions
PIK3R2 5296 VS-5584 CHEMBL1079593 inhibitor ChemblInteractions
PIK3R2 5296 GEDATOLISIB CHEMBL592445 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R2 5296 QUERCETIN CHEMBL50 inhibitor MyCancerGenome
PIK3R2 5296 DACTOLISIB CHEMBL1879463 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R2 5296 TASELISIB CHEMBL2387080 inhibitor ChemblInteractions
PIK3R2 5296 AZD-6482 CHEMBL2165191 inhibitor ChemblInteractions
PIK3R2 5296 Puquitinib CHEMBL3545088 inhibitor ChemblInteractions
PIK3R2 5296 GSK-1059615 CHEMBL3544966 inhibitor ChemblInteractions
PIK3R2 5296 SONOLISIB CHEMBL411907 inhibitor MyCancerGenome, ChemblInteractions, MyCancerGenomeClinicalTrial
PIK3R2 5296 APITOLISIB CHEMBL1922094 inhibitor MyCancerGenome, ChemblInteractions
PIK3R2 5296 PILARALISIB (CHEMBL3360203) CHEMBL3360203 inhibitor ChemblInteractions
PIK3R2 5296 PI-103 CHEMBL573339 inhibitor MyCancerGenome
PIK3R2 5296 ALPELISIB CHEMBL2396661 inhibitor MyCancerGenome, MyCancerGenomeClinicalTrial
PIK3R2 5296 BGT-226 (CHEMBL3545096) CHEMBL3545096 inhibitor ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID