Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
SCN3A 6328 ORPHENADRINE (CHLORIDE) CHEMBL1201023 blocker ChemblInteractions
SCN3A 6328 OXCARBAZEPINE CHEMBL1068 blocker ChemblInteractions
SCN3A 6328 NKTR-171 CHEMBL3545209 blocker ChemblInteractions
SCN3A 6328 NERISPIRDINE CHEMBL2107762 blocker ChemblInteractions
SCN3A 6328 TETRACAINE HYDROCHLORIDE CHEMBL1255654 blocker ChemblInteractions
SCN3A 6328 PRILOCAINE CHEMBL1194 blocker ChemblInteractions
SCN3A 6328 PROPAFENONE HYDROCHLORIDE CHEMBL1201063 blocker ChemblInteractions
SCN3A 6328 LAMOTRIGINE CHEMBL741 blocker ChemblInteractions
SCN3A 6328 ORPHENADRINE CITRATE CHEMBL1200395 blocker ChemblInteractions
SCN3A 6328 MERETHOXYLLINE PROCAINE CHEMBL1200443 blocker ChemblInteractions
SCN3A 6328 DRONEDARONE HYDROCHLORIDE CHEMBL1201729 blocker ChemblInteractions
SCN3A 6328 PROPOXYCAINE HYDROCHLORIDE CHEMBL1769 blocker ChemblInteractions
SCN3A 6328 MEPHENYTOIN CHEMBL861 blocker ChemblInteractions
SCN3A 6328 VERATRIDINE CHEMBL439496 activator GuideToPharmacologyInteractions
SCN3A 6328 SAXITOXIN CHEMBL501134 channel blocker GuideToPharmacologyInteractions
SCN3A 6328 CHEMBL270497 CHEMBL270497 gating inhibitor GuideToPharmacologyInteractions
SCN3A 6328 SAFINAMIDE CHEMBL396778 TdgClinicalTrial
SCN3A 6328 PRIMIDONE CHEMBL856 blocker ChemblInteractions
SCN3A 6328 PROCAINE HYDROCHLORIDE CHEMBL1200841 blocker ChemblInteractions
SCN3A 6328 TOCAINIDE HYDROCHLORIDE CHEMBL1200773 blocker ChemblInteractions
SCN3A 6328 IRAMPANEL CHEMBL29741 blocker ChemblInteractions
SCN3A 6328 ARTICAINE HYDROCHLORIDE CHEMBL1200819 blocker ChemblInteractions
SCN3A 6328 QUINIDINE POLYGALACTURONATE CHEMBL1201486 blocker ChemblInteractions
SCN3A 6328 CHLOROPROCAINE HYDROCHLORIDE CHEMBL944 blocker ChemblInteractions
SCN3A 6328 PHENYTOIN CHEMBL16 blocker ChemblInteractions
SCN3A 6328 RALFINAMIDE CHEMBL2107771 blocker ChemblInteractions
SCN3A 6328 PHENAZOPYRIDINE HYDROCHLORIDE CHEMBL1201022 blocker ChemblInteractions
SCN3A 6328 TETRACAINE CHEMBL698 blocker ChemblInteractions
SCN3A 6328 FOSPHENYTOIN SODIUM CHEMBL919 blocker ChemblInteractions
SCN3A 6328 ZONISAMIDE CHEMBL750 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, DrugBank 19557119, 20025128, 20001433, 18433351, 14704463, 15511691, 19948168
SCN3A 6328 LACOSAMIDE CHEMBL58323 blocker ChemblInteractions, DrugBank 10592235
SCN3A 6328 PHENACEMIDE CHEMBL918 blocker ChemblInteractions
SCN3A 6328 BENOXINATE HYDROCHLORIDE CHEMBL1200654 blocker ChemblInteractions
SCN3A 6328 DISOPYRAMIDE PHOSPHATE CHEMBL1201020 blocker ChemblInteractions
SCN3A 6328 DYCLONINE HYDROCHLORIDE CHEMBL1200478 blocker ChemblInteractions
SCN3A 6328 QUINIDINE SULFATE CHEMBL3707183 blocker ChemblInteractions
SCN3A 6328 TOPIRAMATE CHEMBL220492 blocker ChemblInteractions
SCN3A 6328 ETIDOCAINE HYDROCHLORIDE CHEMBL1200597 blocker ChemblInteractions
SCN3A 6328 INDECAINIDE HYDROCHLORIDE CHEMBL1200341 blocker ChemblInteractions
SCN3A 6328 HEXYLCAINE HYDROCHLORIDE CHEMBL1200715 blocker ChemblInteractions
SCN3A 6328 NW-3509 CHEMBL3545207 blocker ChemblInteractions
SCN3A 6328 ROPIVACAINE HYDROCHLORIDE CHEMBL1889140 blocker ChemblInteractions
SCN3A 6328 MORICIZINE HYDROCHLORIDE CHEMBL1200334 blocker ChemblInteractions
SCN3A 6328 LIDOCAINE HYDROCHLORIDE HYDRATE CHEMBL1200409 blocker ChemblInteractions
SCN3A 6328 RILUZOLE CHEMBL744 blocker ChemblInteractions
SCN3A 6328 ETHOTOIN CHEMBL1095 blocker ChemblInteractions
SCN3A 6328 PHENYTOIN SODIUM CHEMBL1611 blocker ChemblInteractions
SCN3A 6328 CARBAMAZEPINE CHEMBL108 blocker ChemblInteractions
SCN3A 6328 PRILOCAINE HYDROCHLORIDE CHEMBL1200586 blocker ChemblInteractions
SCN3A 6328 ELPETRIGINE CHEMBL29919 blocker ChemblInteractions
SCN3A 6328 ESLICARBAZEPINE CHEMBL315985 blocker ChemblInteractions
SCN3A 6328 PROCAINAMIDE HYDROCHLORIDE CHEMBL605 blocker ChemblInteractions
SCN3A 6328 PROPARACAINE HYDROCHLORIDE CHEMBL1200464 blocker ChemblInteractions
SCN3A 6328 RUFINAMIDE CHEMBL1201754 blocker ChemblInteractions
SCN3A 6328 MEXILETINE HYDROCHLORIDE CHEMBL1200606 blocker ChemblInteractions
SCN3A 6328 ESLICARBAZEPINE ACETATE CHEMBL87992 blocker ChemblInteractions
SCN3A 6328 QUINIDINE GLUCONATE CHEMBL1200437 blocker ChemblInteractions
SCN3A 6328 LIDOCAINE CHEMBL79 blocker ChemblInteractions
SCN3A 6328 MEPIVACAINE HYDROCHLORIDE CHEMBL1200440 blocker ChemblInteractions
SCN3A 6328 TETRODOTOXIN CHEMBL507974 channel blocker TdgClinicalTrial, GuideToPharmacologyInteractions, DrugBank 17663442

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID