Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
SCN5A 6331 PHENACEMIDE CHEMBL918 blocker ChemblInteractions
SCN5A 6331 LIDOCAINE HYDROCHLORIDE HYDRATE CHEMBL1200409 blocker ChemblInteractions
SCN5A 6331 MORICIZINE HYDROCHLORIDE CHEMBL1200334 blocker ChemblInteractions
SCN5A 6331 DIBUCAINE CHEMBL1086 inhibitor, blocker TdgClinicalTrial, TEND, DrugBank, TTD 17139284, 17016423, 11752352, 8798723, 12354567, 9742684
SCN5A 6331 CARBAMAZEPINE CHEMBL108 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 12391287, 17139284, 17016423, 20643904, 20526191
SCN5A 6331 BENZONATATE CHEMBL1374379 antagonist, blocker TdgClinicalTrial, TEND, DrugBank, TTD 23258970
SCN5A 6331 ZONISAMIDE CHEMBL750 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, DrugBank 19557119, 20025128, 20001433, 18433351, 14704463, 15511691, 19948168
SCN5A 6331 ELECLAZINE CHEMBL3707392 inhibitor GuideToPharmacologyInteractions
SCN5A 6331 ROPIVACAINE HYDROCHLORIDE CHEMBL1889140 blocker ChemblInteractions
SCN5A 6331 CHLOROPROCAINE HYDROCHLORIDE CHEMBL944 blocker ChemblInteractions
SCN5A 6331 DYCLONINE HYDROCHLORIDE CHEMBL1200478 blocker ChemblInteractions
SCN5A 6331 MERETHOXYLLINE PROCAINE CHEMBL1200443 blocker ChemblInteractions
SCN5A 6331 PRILOCAINE HYDROCHLORIDE CHEMBL1200586 blocker ChemblInteractions
SCN5A 6331 AZD7009 CHEMBL3545040 blocker ChemblInteractions
SCN5A 6331 TETRACAINE HYDROCHLORIDE CHEMBL1255654 blocker ChemblInteractions
SCN5A 6331 PROPAFENONE CHEMBL631 TdgClinicalTrial, TEND
SCN5A 6331 PRILOCAINE CHEMBL1194 blocker TdgClinicalTrial, ChemblInteractions, TEND, TTD
SCN5A 6331 SAFINAMIDE CHEMBL396778 TdgClinicalTrial
SCN5A 6331 DISOPYRAMIDE CHEMBL517 blocker TdgClinicalTrial, TEND, TTD
SCN5A 6331 FOSPHENYTOIN CHEMBL1201336 blocker TdgClinicalTrial, TEND, TTD
SCN5A 6331 PHENAZOPYRIDINE HYDROCHLORIDE CHEMBL1201022 blocker ChemblInteractions
SCN5A 6331 ARTICAINE HYDROCHLORIDE CHEMBL1200819 blocker ChemblInteractions
SCN5A 6331 MEPIVACAINE HYDROCHLORIDE CHEMBL1200440 blocker ChemblInteractions
SCN5A 6331 NW-3509 CHEMBL3545207 blocker ChemblInteractions
SCN5A 6331 INDECAINIDE CHEMBL1201242 inhibitor, blocker TdgClinicalTrial, TEND, DrugBank, TTD 6206315, 17139284, 17016423, 2476626, 11752352, 2688391
SCN5A 6331 ENCAINIDE CHEMBL315838 inhibitor, blocker TdgClinicalTrial, TEND, DrugBank, TTD 11752352, 1653123, 17016423, 9835260, 16751287
SCN5A 6331 LIDOCAINE CHEMBL79 blocker, channel blocker PharmGKB, TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND
SCN5A 6331 MEXILETINE HYDROCHLORIDE CHEMBL1200606 blocker ChemblInteractions
SCN5A 6331 PRIMIDONE CHEMBL856 blocker ChemblInteractions
SCN5A 6331 PHENYTOIN CHEMBL16 blocker TdgClinicalTrial, ChemblInteractions, TEND
SCN5A 6331 ESLICARBAZEPINE CHEMBL315985 blocker TdgClinicalTrial, ChemblInteractions
SCN5A 6331 DIBUCAINE HYDROCHLORIDE CHEMBL1200612 blocker ChemblInteractions
SCN5A 6331 LITHIUM CHEMBL2146126 PharmGKB
SCN5A 6331 LACOSAMIDE CHEMBL58323 blocker ChemblInteractions
SCN5A 6331 DISOPYRAMIDE PHOSPHATE CHEMBL1201020 blocker ChemblInteractions
SCN5A 6331 TOCAINIDE HYDROCHLORIDE CHEMBL1200773 blocker ChemblInteractions
SCN5A 6331 ESLICARBAZEPINE ACETATE CHEMBL87992 blocker ChemblInteractions
SCN5A 6331 TOPIRAMATE CHEMBL220492 blocker ChemblInteractions
SCN5A 6331 PHENYTOIN SODIUM CHEMBL1611 blocker ChemblInteractions
SCN5A 6331 HEXYLCAINE HYDROCHLORIDE CHEMBL1200715 blocker ChemblInteractions
SCN5A 6331 DRONEDARONE HYDROCHLORIDE CHEMBL1201729 blocker ChemblInteractions
SCN5A 6331 ORPHENADRINE (CHLORIDE) CHEMBL1201023 blocker ChemblInteractions
SCN5A 6331 MEXILETINE CHEMBL558 inhibitor, blocker PharmGKB, TdgClinicalTrial, TEND, DrugBank, TTD 11196553, 11752352, 16168489, 12604879, 12650887, 12123767, 12676070
SCN5A 6331 MORICIZINE CHEMBL1075 inhibitor, blocker TdgClinicalTrial, TEND, DrugBank, TTD 11752352, 17139284, 17016423, 12402511
SCN5A 6331 ETHOTOIN CHEMBL1095 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, TEND, DrugBank, TTD 15066664, 17139284, 17016423, 11752352
SCN5A 6331 FLECAINIDE CHEMBL652 inhibitor, blocker PharmGKB, TdgClinicalTrial, TEND, DrugBank, TTD 11196553, 11307783, 11752352, 10961955, 10617684, 10758053, 15272045, 11535580, 12601084
SCN5A 6331 AJMALINE CHEMBL2105617 inhibitor DrugBank 20174578, 21126620, 20022821, 18599870, 6088360, 20870038
SCN5A 6331 ACONITINE CHEMBL2103747 activator GuideToPharmacologyInteractions
SCN5A 6331 CHEMBL270497 CHEMBL270497 gating inhibitor GuideToPharmacologyInteractions
SCN5A 6331 QUINIDINE SULFATE CHEMBL3707183 blocker ChemblInteractions
SCN5A 6331 ORPHENADRINE CITRATE CHEMBL1200395 blocker ChemblInteractions
SCN5A 6331 INDECAINIDE HYDROCHLORIDE CHEMBL1200341 blocker ChemblInteractions
SCN5A 6331 IRAMPANEL CHEMBL29741 blocker ChemblInteractions
SCN5A 6331 PROCAINAMIDE CHEMBL640 blocker PharmGKB, TdgClinicalTrial, TEND, TTD
SCN5A 6331 DYCLONINE CHEMBL1201217 blocker TTD
SCN5A 6331 QUINIDINE POLYGALACTURONATE CHEMBL1201486 blocker ChemblInteractions
SCN5A 6331 TETRACAINE CHEMBL698 blocker ChemblInteractions
SCN5A 6331 PROPAFENONE HYDROCHLORIDE CHEMBL1201063 blocker ChemblInteractions
SCN5A 6331 PROPOXYCAINE HYDROCHLORIDE CHEMBL1769 blocker ChemblInteractions
SCN5A 6331 ETIDOCAINE HYDROCHLORIDE CHEMBL1200597 blocker ChemblInteractions
SCN5A 6331 TETRODOTOXIN CHEMBL507974 blocker TdgClinicalTrial, TTD
SCN5A 6331 LAMOTRIGINE CHEMBL741 blocker ChemblInteractions
SCN5A 6331 RALFINAMIDE CHEMBL2107771 blocker ChemblInteractions
SCN5A 6331 HEXYLCAINE CHEMBL1197 inhibitor, blocker TdgClinicalTrial, TEND, DrugBank, TTD 11752352, 17139284, 17016423
SCN5A 6331 RANOLAZINE CHEMBL1404 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 19077543, 17220471
SCN5A 6331 MEPHENYTOIN CHEMBL861 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, TEND, DrugBank, TTD 15066664, 11752352, 15001403
SCN5A 6331 RILUZOLE CHEMBL744 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, DrugBank 9262334, 17139284, 17016423, 12440368, 20590601
SCN5A 6331 OXCARBAZEPINE CHEMBL1068 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 17139284, 17016423, 20502724
SCN5A 6331 TOCAINIDE CHEMBL1762 inhibitor, blocker TdgClinicalTrial, TEND, DrugBank, TTD 11752352, 10953551
SCN5A 6331 BENOXINATE HYDROCHLORIDE CHEMBL1200654 blocker ChemblInteractions
SCN5A 6331 QUINIDINE GLUCONATE CHEMBL1200437 blocker ChemblInteractions
SCN5A 6331 PROCAINE HYDROCHLORIDE CHEMBL1200841 blocker ChemblInteractions
SCN5A 6331 NKTR-171 CHEMBL3545209 blocker ChemblInteractions
SCN5A 6331 AZD1305 CHEMBL3545169 blocker ChemblInteractions
SCN5A 6331 FLECAINIDE ACETATE CHEMBL1200822 blocker ChemblInteractions
SCN5A 6331 PROCAINAMIDE HYDROCHLORIDE CHEMBL605 blocker ChemblInteractions
SCN5A 6331 PROPARACAINE HYDROCHLORIDE CHEMBL1200464 blocker ChemblInteractions
SCN5A 6331 BEPRIDIL CHEMBL1008 TdgClinicalTrial, TEND
SCN5A 6331 PROPARACAINE CHEMBL1196 blocker TTD
SCN5A 6331 LICARBAZEPINE CHEMBL1067 TdgClinicalTrial
SCN5A 6331 NERISPIRDINE CHEMBL2107762 blocker ChemblInteractions
SCN5A 6331 RUFINAMIDE CHEMBL1201754 blocker ChemblInteractions
SCN5A 6331 FOSPHENYTOIN SODIUM CHEMBL919 blocker ChemblInteractions
SCN5A 6331 APRINDINE CHEMBL1213033 inhibitor TdgClinicalTrial, DrugBank 1660104, 1653644
SCN5A 6331 COCAINE CHEMBL370805 inhibitor PharmGKB, TdgClinicalTrial, TEND, DrugBank 9876137, 15880981, 17038146
SCN5A 6331 VERAPAMIL CHEMBL6966 other DrugBank 15944809

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID