Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
SCN8A 6334 ETIDOCAINE HYDROCHLORIDE CHEMBL1200597 blocker ChemblInteractions
SCN8A 6334 NW-3509 CHEMBL3545207 blocker ChemblInteractions
SCN8A 6334 VERATRIDINE CHEMBL439496 activator GuideToPharmacologyInteractions
SCN8A 6334 PHENYTOIN SODIUM CHEMBL1611 blocker ChemblInteractions
SCN8A 6334 PROPOXYCAINE HYDROCHLORIDE CHEMBL1769 blocker ChemblInteractions
SCN8A 6334 FOSPHENYTOIN SODIUM CHEMBL919 blocker ChemblInteractions
SCN8A 6334 TETRACAINE HYDROCHLORIDE CHEMBL1255654 blocker ChemblInteractions
SCN8A 6334 TETRACAINE CHEMBL698 blocker ChemblInteractions
SCN8A 6334 PHENYTOIN CHEMBL16 blocker ChemblInteractions
SCN8A 6334 CHLOROPROCAINE HYDROCHLORIDE CHEMBL944 blocker ChemblInteractions
SCN8A 6334 PRIMIDONE CHEMBL856 blocker ChemblInteractions
SCN8A 6334 DISOPYRAMIDE PHOSPHATE CHEMBL1201020 blocker ChemblInteractions
SCN8A 6334 PROCAINE HYDROCHLORIDE CHEMBL1200841 blocker ChemblInteractions
SCN8A 6334 MORICIZINE HYDROCHLORIDE CHEMBL1200334 blocker ChemblInteractions
SCN8A 6334 ORPHENADRINE (CHLORIDE) CHEMBL1201023 blocker ChemblInteractions
SCN8A 6334 LIDOCAINE CHEMBL79 blocker ChemblInteractions
SCN8A 6334 ZONISAMIDE CHEMBL750 blocker ChemblInteractions
SCN8A 6334 ESLICARBAZEPINE ACETATE CHEMBL87992 blocker ChemblInteractions
SCN8A 6334 NKTR-171 CHEMBL3545209 blocker ChemblInteractions
SCN8A 6334 IRAMPANEL CHEMBL29741 blocker ChemblInteractions
SCN8A 6334 INDECAINIDE HYDROCHLORIDE CHEMBL1200341 blocker ChemblInteractions
SCN8A 6334 ARTICAINE HYDROCHLORIDE CHEMBL1200819 blocker ChemblInteractions
SCN8A 6334 RUFINAMIDE CHEMBL1201754 blocker ChemblInteractions
SCN8A 6334 CARBAMAZEPINE CHEMBL108 blocker ChemblInteractions
SCN8A 6334 PHENACEMIDE CHEMBL918 blocker ChemblInteractions
SCN8A 6334 HEXYLCAINE HYDROCHLORIDE CHEMBL1200715 blocker ChemblInteractions
SCN8A 6334 CHEMBL270497 CHEMBL270497 gating inhibitor GuideToPharmacologyInteractions
SCN8A 6334 RILUZOLE CHEMBL744 blocker ChemblInteractions
SCN8A 6334 ETHOTOIN CHEMBL1095 blocker ChemblInteractions
SCN8A 6334 DRONEDARONE HYDROCHLORIDE CHEMBL1201729 blocker ChemblInteractions
SCN8A 6334 QUINIDINE SULFATE CHEMBL3707183 blocker ChemblInteractions
SCN8A 6334 MERETHOXYLLINE PROCAINE CHEMBL1200443 blocker ChemblInteractions
SCN8A 6334 OXCARBAZEPINE CHEMBL1068 blocker ChemblInteractions
SCN8A 6334 LAMOTRIGINE CHEMBL741 blocker ChemblInteractions
SCN8A 6334 LIDOCAINE HYDROCHLORIDE HYDRATE CHEMBL1200409 blocker ChemblInteractions
SCN8A 6334 NERISPIRDINE CHEMBL2107762 blocker ChemblInteractions
SCN8A 6334 LACOSAMIDE CHEMBL58323 blocker ChemblInteractions
SCN8A 6334 SAFINAMIDE CHEMBL396778 TdgClinicalTrial
SCN8A 6334 BENOXINATE HYDROCHLORIDE CHEMBL1200654 blocker ChemblInteractions
SCN8A 6334 PHENAZOPYRIDINE HYDROCHLORIDE CHEMBL1201022 blocker ChemblInteractions
SCN8A 6334 DYCLONINE HYDROCHLORIDE CHEMBL1200478 blocker ChemblInteractions
SCN8A 6334 MEPHENYTOIN CHEMBL861 blocker ChemblInteractions
SCN8A 6334 MEPIVACAINE HYDROCHLORIDE CHEMBL1200440 blocker ChemblInteractions
SCN8A 6334 ORPHENADRINE CITRATE CHEMBL1200395 blocker ChemblInteractions
SCN8A 6334 SAXITOXIN CHEMBL501134 channel blocker GuideToPharmacologyInteractions
SCN8A 6334 MEXILETINE HYDROCHLORIDE CHEMBL1200606 blocker ChemblInteractions
SCN8A 6334 QUINIDINE GLUCONATE CHEMBL1200437 blocker ChemblInteractions
SCN8A 6334 PRILOCAINE CHEMBL1194 blocker ChemblInteractions
SCN8A 6334 TOPIRAMATE CHEMBL220492 blocker ChemblInteractions
SCN8A 6334 PRILOCAINE HYDROCHLORIDE CHEMBL1200586 blocker ChemblInteractions
SCN8A 6334 TOCAINIDE HYDROCHLORIDE CHEMBL1200773 blocker ChemblInteractions
SCN8A 6334 RALFINAMIDE CHEMBL2107771 blocker ChemblInteractions
SCN8A 6334 ESLICARBAZEPINE CHEMBL315985 blocker ChemblInteractions
SCN8A 6334 PROCAINAMIDE HYDROCHLORIDE CHEMBL605 blocker ChemblInteractions
SCN8A 6334 ROPIVACAINE HYDROCHLORIDE CHEMBL1889140 blocker ChemblInteractions
SCN8A 6334 PROPARACAINE HYDROCHLORIDE CHEMBL1200464 blocker ChemblInteractions
SCN8A 6334 QUINIDINE POLYGALACTURONATE CHEMBL1201486 blocker ChemblInteractions
SCN8A 6334 PROPAFENONE HYDROCHLORIDE CHEMBL1201063 blocker ChemblInteractions
SCN8A 6334 TETRODOTOXIN CHEMBL507974 TdgClinicalTrial, DrugBank 17663442

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID
SCN8A rs4512905 TT lithium efficacy no A trend was seen for an association but this did not reach statistical significance for quantitative trait analysis of long-term treatment response scale. Genotype TT is not associated with increased response to lithium in people with Bipolar Disorder as compared to genotype CC. 21961650 827816731