Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
SCN10A 6336 BENZOCAINE CHEMBL278172 inhibitor TdgClinicalTrial, TEND, DrugBank 16174788, 19661462, 17139284, 17016423, 17967784
SCN10A 6336 TETRACAINE CHEMBL698 inhibitor, blocker ChemblInteractions, TTD
SCN10A 6336 ROPIVACAINE HYDROCHLORIDE CHEMBL1889140 blocker ChemblInteractions
SCN10A 6336 BENOXINATE HYDROCHLORIDE CHEMBL1200654 blocker ChemblInteractions
SCN10A 6336 ESLICARBAZEPINE ACETATE CHEMBL87992 blocker ChemblInteractions
SCN10A 6336 NW-3509 CHEMBL3545207 blocker ChemblInteractions
SCN10A 6336 DSP-2230 CHEMBL3545012 blocker ChemblInteractions
SCN10A 6336 Afacifenacin CHEMBL3545165 blocker ChemblInteractions
SCN10A 6336 MEPHENYTOIN CHEMBL861 blocker ChemblInteractions
SCN10A 6336 RANOLAZINE CHEMBL1404 blocker TTD
SCN10A 6336 MEPIVACAINE CHEMBL1087 TdgClinicalTrial, TEND
SCN10A 6336 PHENAZOPYRIDINE HYDROCHLORIDE CHEMBL1201022 blocker ChemblInteractions
SCN10A 6336 ETHOTOIN CHEMBL1095 blocker ChemblInteractions
SCN10A 6336 PROPAFENONE HYDROCHLORIDE CHEMBL1201063 blocker ChemblInteractions
SCN10A 6336 RUFINAMIDE CHEMBL1201754 blocker ChemblInteractions
SCN10A 6336 MERETHOXYLLINE PROCAINE CHEMBL1200443 blocker ChemblInteractions
SCN10A 6336 DIBUCAINE CHEMBL1086 inhibitor TdgClinicalTrial, TEND, DrugBank 8798723, 17139284, 17016423, 9742684
SCN10A 6336 PROCAINE CHEMBL569 inhibitor TdgClinicalTrial, TEND, DrugBank 17139284, 17016423, 2167458, 9768788, 8581044
SCN10A 6336 RILUZOLE CHEMBL744 blocker ChemblInteractions
SCN10A 6336 DRONEDARONE HYDROCHLORIDE CHEMBL1201729 blocker ChemblInteractions
SCN10A 6336 TOPIRAMATE CHEMBL220492 blocker ChemblInteractions
SCN10A 6336 PROCAINE HYDROCHLORIDE CHEMBL1200841 blocker ChemblInteractions
SCN10A 6336 PROPOXYCAINE HYDROCHLORIDE CHEMBL1769 blocker ChemblInteractions
SCN10A 6336 LAMOTRIGINE CHEMBL741 blocker ChemblInteractions
SCN10A 6336 NKTR-171 CHEMBL3545209 blocker ChemblInteractions
SCN10A 6336 ORPHENADRINE CITRATE CHEMBL1200395 blocker ChemblInteractions
SCN10A 6336 ROPIVACAINE CHEMBL1077896 TdgClinicalTrial, TEND
SCN10A 6336 CHLOROPROCAINE CHEMBL1179047 TdgClinicalTrial, TEND
SCN10A 6336 PRILOCAINE HYDROCHLORIDE CHEMBL1200586 blocker ChemblInteractions
SCN10A 6336 DYCLONINE HYDROCHLORIDE CHEMBL1200478 blocker ChemblInteractions
SCN10A 6336 QUINIDINE SULFATE CHEMBL3707183 blocker ChemblInteractions
SCN10A 6336 PF-04531083 CHEMBL3544951 blocker ChemblInteractions
SCN10A 6336 PHENYTOIN CHEMBL16 blocker ChemblInteractions
SCN10A 6336 LIDOCAINE CHEMBL79 blocker TdgClinicalTrial, ChemblInteractions, TEND
SCN10A 6336 PROPARACAINE HYDROCHLORIDE CHEMBL1200464 blocker ChemblInteractions
SCN10A 6336 PROPARACAINE CHEMBL1196 TdgClinicalTrial, TEND
SCN10A 6336 DYCLONINE CHEMBL1201217 inhibitor TdgClinicalTrial, TEND, DrugBank 17139284, 17016423, 9476974, 10355012
SCN10A 6336 COCAINE CHEMBL370805 inhibitor TdgClinicalTrial, TEND, DrugBank 17139284, 17016423
SCN10A 6336 LACOSAMIDE CHEMBL58323 blocker ChemblInteractions, DrugBank 10592235
SCN10A 6336 PHENACEMIDE CHEMBL918 blocker ChemblInteractions
SCN10A 6336 HEXYLCAINE HYDROCHLORIDE CHEMBL1200715 blocker ChemblInteractions
SCN10A 6336 MORICIZINE HYDROCHLORIDE CHEMBL1200334 blocker ChemblInteractions
SCN10A 6336 ETIDOCAINE HYDROCHLORIDE CHEMBL1200597 blocker ChemblInteractions
SCN10A 6336 OXCARBAZEPINE CHEMBL1068 blocker ChemblInteractions
SCN10A 6336 LIDOCAINE HYDROCHLORIDE HYDRATE CHEMBL1200409 blocker ChemblInteractions
SCN10A 6336 TOCAINIDE HYDROCHLORIDE CHEMBL1200773 blocker ChemblInteractions
SCN10A 6336 ZONISAMIDE CHEMBL750 blocker ChemblInteractions
SCN10A 6336 NERISPIRDINE CHEMBL2107762 blocker ChemblInteractions
SCN10A 6336 RALFINAMIDE CHEMBL2107771 blocker ChemblInteractions
SCN10A 6336 TETRACAINE HYDROCHLORIDE CHEMBL1255654 blocker ChemblInteractions
SCN10A 6336 DIBUCAINE HYDROCHLORIDE CHEMBL1200612 blocker ChemblInteractions
SCN10A 6336 MEPIVACAINE HYDROCHLORIDE CHEMBL1200440 blocker ChemblInteractions
SCN10A 6336 PROCAINAMIDE HYDROCHLORIDE CHEMBL605 blocker ChemblInteractions
SCN10A 6336 BUPIVACAINE CHEMBL1098 TdgClinicalTrial, TEND
SCN10A 6336 TIAPRIDE CHEMBL84158 inhibitor TTD
SCN10A 6336 PRIMIDONE CHEMBL856 blocker ChemblInteractions
SCN10A 6336 ESLICARBAZEPINE CHEMBL315985 blocker ChemblInteractions
SCN10A 6336 DISOPYRAMIDE PHOSPHATE CHEMBL1201020 blocker ChemblInteractions
SCN10A 6336 PHENYTOIN SODIUM CHEMBL1611 blocker ChemblInteractions
SCN10A 6336 HEXYLCAINE CHEMBL1197 inhibitor TdgClinicalTrial, TEND, DrugBank 17139284, 17016423
SCN10A 6336 BENOXINATE CHEMBL1200 inhibitor TdgClinicalTrial, TEND, DrugBank 19429093, 17139284, 17016423
SCN10A 6336 LEVOBUPIVACAINE CHEMBL1201193 inhibitor TdgClinicalTrial, TEND, DrugBank 11094008, 17139284, 17016423, 10969308, 16418020
SCN10A 6336 QUINIDINE POLYGALACTURONATE CHEMBL1201486 blocker ChemblInteractions
SCN10A 6336 CHLOROPROCAINE HYDROCHLORIDE CHEMBL944 blocker ChemblInteractions
SCN10A 6336 MEXILETINE HYDROCHLORIDE CHEMBL1200606 blocker ChemblInteractions
SCN10A 6336 QUINIDINE GLUCONATE CHEMBL1200437 blocker ChemblInteractions
SCN10A 6336 PRILOCAINE CHEMBL1194 blocker ChemblInteractions
SCN10A 6336 ORPHENADRINE (CHLORIDE) CHEMBL1201023 blocker ChemblInteractions
SCN10A 6336 FOSPHENYTOIN SODIUM CHEMBL919 blocker ChemblInteractions
SCN10A 6336 INDECAINIDE HYDROCHLORIDE CHEMBL1200341 blocker ChemblInteractions
SCN10A 6336 ARTICAINE HYDROCHLORIDE CHEMBL1200819 blocker ChemblInteractions
SCN10A 6336 CARBAMAZEPINE CHEMBL108 blocker ChemblInteractions
SCN10A 6336 TETRODOTOXIN CHEMBL507974 TdgClinicalTrial
SCN10A 6336 IRAMPANEL CHEMBL29741 blocker ChemblInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID