Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
BRAF 673 VEMURAFENIB CHEMBL1229517 inhibitor DrugBank, TdgClinicalTrial, CGI, ChemblInteractions, GuideToPharmacologyInteractions, OncoKB, TTD, PharmGKB, CancerCommons, MyCancerGenomeClinicalTrial, ClearityFoundationClinicalTrial, MyCancerGenome, FDA, TALC, ClearityFoundationBiomarkers, CIViC, CKB, DoCM 22743296, 22621641, 23612012, 22608338, 20818844, 23489023, 23288408, 231718, 23094782, 27080216, 26776917, 25466451, 26287849, 23733758, 26200454, 24888229, 25089220, 19884556, 20619739, 19001320, 23617957, 22448344, 22735384, 23846731, 25265494, 25287827, 25399551, 23051966, 23918947, 22663011, 25265492, 24508103, 23020132, 24576830, 22281684, 21639808, 22356324, 24987354, 27048246, 27460442, 24997557, 27729313, 24345920, 23715574, 26989536, 22798288, 24112705, 25515853, 28783719, 26343583, 27523909, 24283590, 26343582, 21107323, 26352686, 25665005, 27297867, 25589621, 23365119, 28649441, 26918217, 27312529, 26460303, 26603897, 27048951, 24523613, 22389471, 25939769, 26267534, 21383288, 24448821, 28514312, 26137449, 24035431, 26732095, 25706985, 24265153, 26582644, 27760111, 26984758, 27500726, 27196754, 24265152, 12068308, 12460919, 21483012, 22773810, 25989278, 25157968, 23934108, 22805292, 21683865, 23549875, 15035987, 21594703, 24354346, 21163703, 24586605, 26619011, 22241789, 24107445, 20368568, 24583796, 24396464, 22972589, 22649091, 23614898, 23812671, 20413299, 21426297, 20630094, 24570209, 25370471, 19404918, 23524406, 19238210, 22997239, 23833300, 22048237, 22351686, 23031422, 19255327, 19561230, 24163374, 20350999, 25024077, 26678033, 21975775, 19537845, 20857202, 19010912, 24388723, 23325582, 22586120, 19018267, 24594804, 23251002, 23470635, 22536370, 21129611, 23406027, 18541894, 12460918, 21663470, 21156289, 22180495, 14679157, 23845441, 19773371, 22038996, 25656898
BRAF 673 PANITUMUMAB CHEMBL1201827 OncoKB, CKB, CGI, CIViC, DoCM 20619739, 21163703, 23325582, 12068308, 22743296, 12460919, 21483012, 22608338, 22773810, 20818844, 25989278, 25157968, 23934108, 22805292, 21683865, 23549875, 22663011, 15035987, 21594703, 24354346, 23918947, 24586605, 26619011, 22241789, 24107445, 19001320, 20368568, 24583796, 24396464, 22972589, 22649091, 23614898, 23812671, 20413299, 21639808, 21426297, 23489023, 20630094, 23612012, 24570209, 25370471, 19404918, 22281684, 22735384, 23524406, 19238210, 22997239, 23020132, 22389471, 24576830, 23833300, 22048237, 22351686, 23031422, 19255327, 19561230, 24163374, 20350999, 25024077, 22448344, 26678033, 21975775, 19537845, 20857202, 24508103, 19010912, 24388723, 22586120, 19018267, 24594804, 23251002, 23470635, 22536370, 21129611, 23406027, 18541894, 12460918, 22356324, 21663470, 21156289, 22180495, 14679157, 23845441, 19773371, 22038996, 19884556, 23617957, 25673644, 25589621, 28514312, 27312529, 28783719, 27770002
BRAF 673 CHEMBL523411 CHEMBL523411 inhibitor TdgClinicalTrial, ClearityFoundationClinicalTrial, MyCancerGenomeClinicalTrial, TTD
BRAF 673 PIMASERTIB CHEMBL2107832 ClearityFoundationBiomarkers, CKB 23629727
BRAF 673 CRIZOTINIB CHEMBL601719 CGI
BRAF 673 PICTILISIB CHEMBL521851 CKB, CIViC 23845441, 19276360, 24265153, 26577700
BRAF 673 DACTOLISIB CHEMBL1879463 CKB, CIViC 23549875, 26137449
BRAF 673 EVEROLIMUS CHEMBL1908360 CKB 27217440, 27797976, 23629727, 20664174, 20664172
BRAF 673 LEUCOVORIN CHEMBL1679 CKB 27626067
BRAF 673 ERLOTINIB CHEMBL553 CKB 27924459, 22448344, 27659046
BRAF 673 IDELALISIB CHEMBL2216870 CKB 26137449
BRAF 673 VENETOCLAX CHEMBL3137309 CKB 27974663
BRAF 673 CAPMATINIB CHEMBL3188267 CKB 28783719
BRAF 673 UPROSERTIB CHEMBL3137336 CKB 24265152
BRAF 673 ATEZOLIZUMAB CHEMBL3707227 CKB
BRAF 673 BEVACIZUMAB CHEMBL1201583 CKB 21216929
BRAF 673 SELUMETINIB CHEMBL1614701 ClearityFoundationBiomarkers, OncoKB, CKB, CGI 26324360, 26343583, 22048237, 27217440, 19915144, 27312529, 27222538, 26461489, 23942066, 24448821, 22197931, 26137449, 27655129, 23406027, 26351322, 27196754, 24265152
BRAF 673 DABRAFENIB CHEMBL2028663 inhibitor CGI, GuideToPharmacologyInteractions, DrugBank, OncoKB, MyCancerGenome, TALC, CancerCommons, CIViC, CKB, DoCM 26392102, 2015, 8006, 23524406, 22608338, 2013, 8009, 2014, 38, 20818844, 23489023, 27080216, 23470635, 23621583, 22743296, 26776917, 25466451, 26287849, 23733758, 26200454, 24888229, 25089220, 19884556, 20619739, 19001320, 23617957, 22448344, 22663011, 27283860, 22735384, 23846731, 25265494, 25287827, 25399551, 23051966, 23918947, 25265492, 24508103, 23020132, 23463675, 24583796, 27048246, 23031422, 25673644, 27577079, 27523909, 25370473, 27797976, 22389471, 27312529, 24885690, 28268064, 28784858, 27697975, 24265154, 24265153, 28891408, 27255157, 26732095, 27770002, 27659046, 27500726, 26811525, 28512244, 12068308, 12460919, 21483012, 22773810, 25989278, 25157968, 23934108, 22805292, 21683865, 23549875, 15035987, 21594703, 24354346, 21163703, 24586605, 26619011, 22241789, 24107445, 20368568, 24396464, 22972589, 22649091, 23614898, 23812671, 20413299, 21639808, 21426297, 20630094, 23612012, 24570209, 25370471, 19404918, 22281684, 19238210, 22997239, 24576830, 23833300, 22048237, 22351686, 19255327, 19561230, 24163374, 20350999, 25024077, 26678033, 21975775, 19537845, 20857202, 19010912, 24388723, 23325582, 22586120, 19018267, 24594804, 23251002, 22536370, 21129611, 23406027, 18541894, 12460918, 22356324, 21663470, 21156289, 22180495, 14679157, 23845441, 19773371, 22038996, 25656898
BRAF 673 CHEMBL525191 CHEMBL525191 inhibitor CKB, GuideToPharmacologyInteractions, CIViC 19276360, 23549875
BRAF 673 SB590885 CHEMBL477989 inhibitor CKB, GuideToPharmacologyInteractions 20538618, 27523909
BRAF 673 SORAFENIB CHEMBL1336 inhibitor OncoKB, TdgClinicalTrial, CGI, GuideToPharmacologyInteractions, DrugBank, MyCancerGenome, TTD, MyCancerGenomeClinicalTrial, ClearityFoundationClinicalTrial, TEND, CIViC, CKB, DoCM 23152448, 20586710, 20332142, 25662396, 15466206, 24422672, 238900088, 20526349, 24727320, 16880785, 16901402, 11752352, 17575107, 16609060, 20812347, 19001320, 20538618, 27388325, 23629727, 22394203, 23792568, 24885690, 26619011, 21129611, 14679157, 20619739, 12068308, 19537845, 20350999, 22310681, 25157968, 18794803, 18186519
BRAF 673 XL-281 CHEMBL3545027 inhibitor MyCancerGenome, TdgClinicalTrial, ChemblInteractions, DrugBank, TTD
BRAF 673 CHEMBL526479 CHEMBL526479 DrugBank 10592235
BRAF 673 CETUXIMAB CHEMBL1201577 OncoKB, CKB, CGI, CIViC, DoCM 20619739, 21163703, 23325582, 19884556, 19001320, 23617957, 22448344, 22281684, 27729313, 25714871, 27002107, 25838391, 27312529, 26916115, 26208524, 24523613, 22270724, 28783719, 28363909, 26287849, 12068308, 22743296, 12460919, 21483012, 22608338, 22773810, 20818844, 25989278, 25157968, 23934108, 22805292, 21683865, 23549875, 22663011, 15035987, 21594703, 24354346, 23918947, 24586605, 26619011, 22241789, 24107445, 20368568, 24583796, 24396464, 22972589, 22649091, 23614898, 23812671, 20413299, 21639808, 21426297, 23489023, 20630094, 23612012, 24570209, 25370471, 19404918, 22735384, 23524406, 19238210, 22997239, 23020132, 22389471, 24576830, 23833300, 22048237, 22351686, 23031422, 19255327, 19561230, 24163374, 20350999, 25024077, 26678033, 21975775, 19537845, 20857202, 24508103, 19010912, 24388723, 22586120, 19018267, 24594804, 23251002, 23470635, 22536370, 21129611, 23406027, 18541894, 12460918, 22356324, 21663470, 21156289, 22180495, 14679157, 23845441, 19773371, 22038996
BRAF 673 TEMSIROLIMUS CHEMBL1201182 inhibitor OncoKB, CKB, MyCancerGenomeClinicalTrial 21216929, 23152448, 20586710, 20332142, 25662396, 15466206, 24422672
BRAF 673 DABRAFENIB MESYLATE CHEMBL2105729 inhibitor ChemblInteractions, MyCancerGenomeClinicalTrial
BRAF 673 MLN-2480 CHEMBL3348923 inhibitor CKB, ChemblInteractions, MyCancerGenomeClinicalTrial
BRAF 673 ALPELISIB CHEMBL2396661 CKB, CGI 27312529, 28363909, 26577700, 27924459, 27659046
BRAF 673 GEFITINIB CHEMBL939 CKB, CIViC 22281684, 22448344, 23242808, 27312529
BRAF 673 BUPARLISIB CHEMBL2017974 CKB 27307593, 24265152
BRAF 673 PALBOCICLIB CHEMBL189963 CKB 27488531, 26369631
BRAF 673 TRASTUZUMAB CHEMBL1201585 CKB 27626067
BRAF 673 BI-2536 CHEMBL513909 CKB 26573800
BRAF 673 GEDATOLISIB CHEMBL592445 CKB 24042735, 21325073, 17314276
BRAF 673 GSK-2636771 CHEMBL3188551 CKB 26645196, 26577700
BRAF 673 PHENMETRAZINE CHEMBL1201208 CKB 26137449
BRAF 673 Voruciclib CHEMBL3545218 CKB
BRAF 673 TUBASTATIN A CHEMBL2018302 CKB 25957812
BRAF 673 LGX-806 CHEMBL3545263 inhibitor ChemblInteractions
BRAF 673 BGB-283 CHEMBL3545246 inhibitor CKB, GuideToPharmacologyInteractions, ChemblInteractions 26208524
BRAF 673 CHIR-265 CHEMBL558752 inhibitor MyCancerGenome, TdgClinicalTrial, CKB, GuideToPharmacologyInteractions, ChemblInteractions, CancerCommons 22351689, 20538618
BRAF 673 LY-3009120 CHEMBL3545195 inhibitor CKB, GuideToPharmacologyInteractions, ChemblInteractions, CIViC 26732095, 26343583, 22798288
BRAF 673 PLX-8394 CHEMBL3545005 inhibitor CKB, GuideToPharmacologyInteractions, ChemblInteractions 24422853, 27834212
BRAF 673 ENCORAFENIB CHEMBL3301612 inhibitor TALC, MyCancerGenome, OncoKB, CKB, ChemblInteractions, CancerCommons 27312529, 26577700, 28363909, 19884556, 20619739, 19001320, 23617957, 22448344, 28351928, 27307593
BRAF 673 BINIMETINIB CHEMBL3187723 ClearityFoundationBiomarkers, OncoKB, CKB 19884556, 20619739, 19001320, 23617957, 22448344, 27307593, 23414587, 26577700, 28152546
BRAF 673 COBIMETINIB CHEMBL2146883 ClearityFoundationBiomarkers, OncoKB, CKB, CGI, CIViC, FDA 22735384, 23846731, 25265494, 25287827, 25399551, 22608338, 23051966, 23918947, 20818844, 22663011, 25265492, 24508103, 23020132, 25089220, 23934108, 28649441, 22084396
BRAF 673 PACLITAXEL CHEMBL428647 OncoKB 26324360
BRAF 673 OMIPALISIB CHEMBL1236962 CKB 22389471
BRAF 673 Ribociclib CHEMBL3545110 CKB 28351928
BRAF 673 ARQ-092 CHEMBL3545422 CKB 26469692
BRAF 673 INK-128 CHEMBL3545056 CKB 25261369, 26272063
BRAF 673 PF-04217903 CHEMBL2001019 CKB 27659046
BRAF 673 NIVOLUMAB CHEMBL2108738 FDA
BRAF 673 CEP-32496 CHEMBL2029988 inhibitor CKB, GuideToPharmacologyInteractions, ChemblInteractions 22319199
BRAF 673 CHEMBL373011 CHEMBL373011 inhibitor GuideToPharmacologyInteractions
BRAF 673 PLX-4720 CHEMBL1230020 inhibitor CKB, GuideToPharmacologyInteractions, CGI, CIViC, DrugBank 10592235, 23845441, 18287029, 20538618, 26573800, 26461489, 27924459, 24983357, 27523909, 23242808, 27217440, 22281684, 19915144, 24265153, 21383288, 26351322
BRAF 673 REGORAFENIB CHEMBL1946170 inhibitor MyCancerGenome, CKB, GuideToPharmacologyInteractions, ChemblInteractions, DrugBank, MyCancerGenomeClinicalTrial 25838391, 23629727, 21170960
BRAF 673 TRAMETINIB CHEMBL2103875 ClearityFoundationBiomarkers, OncoKB, CKB, CGI, CIViC, DoCM, FDA 26392102, 2015, 8006, 23248257, 22805292, 24727320, 24345920, 20526349, 24583796, 25399551, 27048246, 27283860, 23020132, 22663011, 22169769, 24933606, 22798288, 26314551, 27577079, 28783719, 27488531, 27797976, 22389471, 27312529, 25665005, 27297867, 28268064, 27222538, 27697975, 26916115, 25309914, 26469692, 24265153, 24265154, 26369631, 28891408, 25265492, 26732095, 25706985, 25370473, 28344857, 27760111, 27770002, 26343583, 27500726, 26811525, 24265152, 28784858, 27338794, 28512244, 25089220, 26343582, 20141835, 22735384, 23846731, 25265494, 25287827, 22608338, 23051966, 23918947, 20818844, 24508103, 12068308, 22743296, 12460919, 21483012, 22773810, 25989278, 25157968, 23934108, 21683865, 23549875, 15035987, 21594703, 24354346, 21163703, 24586605, 26619011, 22241789, 24107445, 19001320, 20368568, 24396464, 22972589, 22649091, 23614898, 23812671, 20413299, 21639808, 21426297, 23489023, 20630094, 23612012, 24570209, 25370471, 19404918, 22281684, 23524406, 19238210, 22997239, 24576830, 23833300, 22048237, 22351686, 23031422, 19255327, 20619739, 19561230, 24163374, 20350999, 25024077, 22448344, 26678033, 21975775, 19537845, 20857202, 19010912, 24388723, 23325582, 22586120, 19018267, 24594804, 23251002, 23470635, 22536370, 21129611, 23406027, 18541894, 12460918, 22356324, 21663470, 21156289, 22180495, 14679157, 23845441, 19773371, 22038996, 25656898, 23715574, 2493360
BRAF 673 ARQ-736 CHEMBL3545296 inhibitor TALC, MyCancerGenome, ChemblInteractions
BRAF 673 RG-7256 CHEMBL3545080 inhibitor MyCancerGenome, ChemblInteractions, CancerCommons
BRAF 673 DASATINIB CHEMBL1421 inhibitor CKB, CGI, DoCM, MyCancerGenomeClinicalTrial 19010912, 23833300, 12068308, 22649091, 19238210, 21483012, 12460918, 12460919, 26619011, 18186519, 19537845, 25157968, 22310681, 21129611, 20350999, 27222538, 23242808
BRAF 673 SORAFENIB TOSYLATE CHEMBL1200485 inhibitor ChemblInteractions, MyCancerGenomeClinicalTrial
BRAF 673 PD-0325901 CHEMBL507361 ClearityFoundationBiomarkers, CKB 26267534, 16273091, 26573800, 27488531, 26272063
BRAF 673 IRINOTECAN CHEMBL481 CKB, CIViC 27729313, 25714871, 28783719
BRAF 673 TAK-733 CHEMBL1615025 CKB, CIViC 22798288, 24398428, 26439693
BRAF 673 FLUOROURACIL CHEMBL185 CKB 27626067, 26637369
BRAF 673 GANETESPIB CHEMBL2103879 CKB 24398428, 25077897
BRAF 673 NAVITOCLAX CHEMBL443684 CKB 25665005, 24983357, 27659046
BRAF 673 ZSTK-474 CHEMBL586701 CKB 26137449
BRAF 673 AZD-6482 CHEMBL2165191 CKB 26577700
BRAF 673 AEW-541 CHEMBL551064 CKB 26577700
BRAF 673 MK-2206 CHEMBL1079175 CKB 24265152
BRAF 673 NERATINIB CHEMBL180022 CKB 26243863
BRAF 673 AFATINIB CHEMBL1173655 CKB 26916115
BRAF 673 SAR-260301 CHEMBL3545008 CKB 27196754
BRAF 673 CHEMBL2204502 CHEMBL2204502 CKB 22351686
BRAF 673 LAPATINIB CHEMBL554 CKB 21464044, 23365119
BRAF 673 TIVOZANIB CHEMBL1289494 CKB 26461489
BRAF 673 CHEMBL217354 CHEMBL217354 CKB 25665005
BRAF 673 E-6201 CHEMBL1097999 CKB 24448821, 23039341
BRAF 673 CEDIRANIB CHEMBL491473 CKB 26461489
BRAF 673 Refametinib CHEMBL2138601 CKB 19706763
BRAF 673 OXALIPLATIN CHEMBL414804 CKB 26637369
BRAF 673 CHEMBL458997 CHEMBL458997 CKB 26090892
BRAF 673 OBATOCLAX CHEMBL408194 CKB 22460902
BRAF 673 CHEMBL1231206 CHEMBL1231206 CKB 26140595
BRAF 673 PA-799 CHEMBL1684984 CKB 21558396
BRAF 673 PEMBROLIZUMAB CHEMBL3137343 CKB, FDA 26645196
BRAF 673 LENVATINIB CHEMBL1289601 CKB 26169970
BRAF 673 IMATINIB CHEMBL941 CKB 27924459
BRAF 673 PF-00477736 CHEMBL3545137 CKB 26140595
BRAF 673 CI-1040 CHEMBL105442 CKB 20538618, 19915144, 19018267
BRAF 673 PANOBINOSTAT CHEMBL483254 CKB 21464044
BRAF 673 DOXORUBICIN CHEMBL53463 CKB 27924459
BRAF 673 SARACATINIB CHEMBL217092 CKB 23242808
BRAF 673 Ro-4987655 CHEMBL1614766 CKB 26438159
BRAF 673 VORINOSTAT CHEMBL98 CKB 27924459
BRAF 673 PLX-3397 CHEMBL3545158 CKB 25939769
BRAF 673 PILARALISIB (CHEMBL3218575) CHEMBL3218575 CKB 25637314
BRAF 673 LY-294002 CHEMBL98350 CKB 23039341

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID