Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
CACNA1S 779 VERAPAMIL CHEMBL6966 inhibitor TdgClinicalTrial, TEND, DrugBank 19125880
CACNA1S 779 NIFEDIPINE CHEMBL193 inhibitor, blocker ChemblInteractions, DrugBank 16675661
CACNA1S 779 DRONEDARONE HYDROCHLORIDE CHEMBL1201729 blocker ChemblInteractions
CACNA1S 779 DRONEDARONE CHEMBL184412 DrugBank
CACNA1S 779 AZD1305 CHEMBL3545169 blocker ChemblInteractions
CACNA1S 779 AMLODIPINE MALEATE CHEMBL1200984 blocker ChemblInteractions
CACNA1S 779 GABAPENTIN CHEMBL940 modulator ChemblInteractions
CACNA1S 779 NIMODIPINE CHEMBL1428 inhibitor, blocker ChemblInteractions, DrugBank 20661350, 20335610, 17705883, 20334460, 16675661, 19844625
CACNA1S 779 FELODIPINE CHEMBL1480 inhibitor, blocker TdgClinicalTrial, ChemblInteractions, DrugBank 16675661
CACNA1S 779 NITRENDIPINE CHEMBL475534 inhibitor DrugBank 16675661
CACNA1S 779 CLEVIDIPINE CHEMBL1237132 blocker TdgClinicalTrial, ChemblInteractions, DrugBank 15492770
CACNA1S 779 NILVADIPINE CHEMBL517427 inhibitor DrugBank 16675661
CACNA1S 779 AMLODIPINE CHEMBL1491 TdgClinicalTrial
CACNA1S 779 CELECOXIB CHEMBL118 PharmGKB
CACNA1S 779 PREGABALIN CHEMBL1059 modulator ChemblInteractions
CACNA1S 779 ELPETRIGINE CHEMBL29919 blocker ChemblInteractions
CACNA1S 779 VERAPAMIL HYDROCHLORIDE CHEMBL1280 blocker ChemblInteractions
CACNA1S 779 DILTIAZEM MALATE CHEMBL1200805 blocker ChemblInteractions
CACNA1S 779 ISRADIPINE CHEMBL1648 inhibitor, blocker ChemblInteractions, DrugBank 16675661
CACNA1S 779 NISOLDIPINE CHEMBL1726 inhibitor, blocker ChemblInteractions, DrugBank 16675661
CACNA1S 779 CINNARIZINE CHEMBL43064 inhibitor DrugBank 1281221, 3530295
CACNA1S 779 MAGNESIUM SULFATE CHEMBL1200456 DrugBank 17139284, 17016423
CACNA1S 779 BEPRIDIL HYDROCHLORIDE CHEMBL1200382 blocker ChemblInteractions
CACNA1S 779 GABAPENTIN ENACARBIL CHEMBL1628502 modulator ChemblInteractions
CACNA1S 779 ATAGABALIN CHEMBL593430 modulator ChemblInteractions
CACNA1S 779 DILTIAZEM HYDROCHLORIDE CHEMBL1697 blocker ChemblInteractions
CACNA1S 779 IMAGABALIN CHEMBL2103836 modulator ChemblInteractions
CACNA1S 779 AMLODIPINE BESYLATE CHEMBL1200402 blocker ChemblInteractions
CACNA1S 779 NICARDIPINE HYDROCHLORIDE CHEMBL1200326 blocker ChemblInteractions
CACNA1S 779 MIBEFRADIL CHEMBL45816 inhibitor DrugBank 10372226, 16899990, 10665814

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID