Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GABBR2 9568 BACLOFEN CHEMBL701 agonist TdgClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, TEND, DrugBank 11008066, 8388192, 10751439, 10545129, 10328880, 19303900, 10658574, 15235087
GABBR2 9568 CHEMBL40157 CHEMBL40157 antagonist GuideToPharmacologyInteractions
GABBR2 9568 CHEMBL1213187 CHEMBL1213187 antagonist GuideToPharmacologyInteractions
GABBR2 9568 CHEMBL312403 CHEMBL312403 antagonist GuideToPharmacologyInteractions
GABBR2 9568 CHEMBL112797 CHEMBL112797 DrugBank
GABBR2 9568 ARBACLOFEN CHEMBL301742 agonist TdgClinicalTrial, ChemblInteractions, DrugBank 11008066, 8388192, 10751439, 10545129, 10328880, 19303900, 10658574, 15235087
GABBR2 9568 ARBACLOFEN PLACARBIL CHEMBL2107312 agonist ChemblInteractions, DrugBank 11008066, 8388192, 10751439, 10545129, 10328880, 19303900, 10658574, 15235087
GABBR2 9568 Lesogaberan CHEMBL448343 agonist TdgClinicalTrial, ChemblInteractions
GABBR2 9568 GAMMA-AMINOBUTYRIC ACID CHEMBL96 agonist GuideToPharmacologyInteractions
GABBR2 9568 CHEMBL455185 CHEMBL455185 antagonist GuideToPharmacologyInteractions
GABBR2 9568 OXYBATE CHEMBL1342 TdgClinicalTrial
GABBR2 9568 SODIUM OXYBATE CHEMBL1200682 agonist ChemblInteractions
GABBR2 9568 PHACLOFEN CHEMBL1255941 antagonist GuideToPharmacologyInteractions
GABBR2 9568 CHEMBL1895916 CHEMBL1895916 antagonist GuideToPharmacologyInteractions
GABBR2 9568 CHEMBL112203 CHEMBL112203 agonist GuideToPharmacologyInteractions

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID