Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
GRIN3A 116443 ROLICYCLIDINE CHEMBL1719398 DrugBank 20613880, 20641908
GRIN3A 116443 PHENCYCLIDINE CHEMBL275528 antagonist DrugBank 17139284, 17016423
GRIN3A 116443 NERAMEXANE CHEMBL2110954 TdgClinicalTrial, DrugBank
GRIN3A 116443 Indantadol CHEMBL3707400 antagonist TdgClinicalTrial, ChemblInteractions
GRIN3A 116443 CHEMBL334533 CHEMBL334533 TdgClinicalTrial
GRIN3A 116443 AV-101 CHEMBL3545351 antagonist ChemblInteractions
GRIN3A 116443 GW468816 CHEMBL1207366 antagonist ChemblInteractions
GRIN3A 116443 ORPHENADRINE (CHLORIDE) CHEMBL1201023 antagonist ChemblInteractions
GRIN3A 116443 METHADONE CHEMBL651 antagonist DrugBank 17139284, 17016423, 19717013
GRIN3A 116443 PROCAINE CHEMBL569 antagonist DrugBank 17139284, 17016423, 11812692, 16299047
GRIN3A 116443 AMANTADINE HYDROCHLORIDE CHEMBL1569 antagonist ChemblInteractions, DrugBank 15800186, 10443547
GRIN3A 116443 AZD8108 CHEMBL3707355 antagonist ChemblInteractions
GRIN3A 116443 CNS-5161 CHEMBL41306 blocker TdgClinicalTrial, ChemblInteractions
GRIN3A 116443 ESKETAMINE HYDROCHLORIDE CHEMBL2364609 ChemblInteractions
GRIN3A 116443 ORPHENADRINE CHEMBL900 TdgClinicalTrial, TEND
GRIN3A 116443 ACAMPROSATE CHEMBL1201293 TdgClinicalTrial
GRIN3A 116443 ACAMPROSATE CALCIUM CHEMBL2068724 antagonist ChemblInteractions
GRIN3A 116443 ORPHENADRINE CITRATE CHEMBL1200395 antagonist ChemblInteractions
GRIN3A 116443 KETAMINE CHEMBL742 TdgClinicalTrial, TEND
GRIN3A 116443 L-GLUTAMATE CHEMBL575060 DrugBank 17139284, 17016423
GRIN3A 116443 FELBAMATE CHEMBL1094 antagonist TdgClinicalTrial, ChemblInteractions, TEND, DrugBank 17139284, 17016423
GRIN3A 116443 NRX-1074 CHEMBL3545230 partial agonist ChemblInteractions
GRIN3A 116443 RAPASTINEL CHEMBL3544917 partial agonist ChemblInteractions
GRIN3A 116443 RALFINAMIDE CHEMBL2107771 antagonist ChemblInteractions
GRIN3A 116443 ESKETAMINE CHEMBL395091 ChemblInteractions
GRIN3A 116443 MEMANTINE HYDROCHLORIDE CHEMBL1699 ChemblInteractions
GRIN3A 116443 LANICEMINE CHEMBL2107647 blocker TdgClinicalTrial, ChemblInteractions
GRIN3A 116443 MEMANTINE CHEMBL807 TdgClinicalTrial, TEND
GRIN3A 116443 DELUCEMINE CHEMBL2110814 antagonist ChemblInteractions
GRIN3A 116443 ETHOPROPAZINE CHEMBL1206 antagonist DrugBank 17139284, 17016423, 12681372, 2849655
GRIN3A 116443 HALOTHANE CHEMBL931 antagonist DrugBank 8968191
GRIN3A 116443 TENOCYCLIDINE CHEMBL279676 antagonist DrugBank 17157509, 2538766
GRIN3A 116443 NERAMEXANE MESYLATE CHEMBL2106798 antagonist ChemblInteractions
GRIN3A 116443 LATREPIRDINE CHEMBL589390 TdgClinicalTrial
GRIN3A 116443 DEXTROMETHORPHAN CHEMBL52440 TdgClinicalTrial, TEND
GRIN3A 116443 NEBOGLAMINE CHEMBL1255840 positive allosteric modulator ChemblInteractions
GRIN3A 116443 KETAMINE HYDROCHLORIDE CHEMBL1714 ChemblInteractions
GRIN3A 116443 ACETYLCYSTEINE CHEMBL600 activator DrugBank 12183209

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID