Gene-drug interactions (data source: DGIdb)
Gene Name Entrez ID Drug Name Chembl ID Interaction Types Sources publications
MAP2K1 5604 COBIMETINIB CHEMBL2146883 inhibitor, allosteric modulator OncoKB, ChemblInteractions, TALC, DrugBank, GuideToPharmacologyInteractions, CancerCommons, TdgClinicalTrial, MyCancerGenome, ClearityFoundationClinicalTrial, MyCancerGenomeClinicalTrial, CKB 23846731, 25351745, 22663011, 26324360, 26566875, 25370473, 26384788
MAP2K1 5604 K-252A CHEMBL281948 DrugBank 10592235
MAP2K1 5604 LEUCOVORIN CHEMBL1679 inhibitor GuideToPharmacologyInteractions
MAP2K1 5604 PIMASERTIB CHEMBL2107832 inhibitor TALC, MyCancerGenome, ClearityFoundationClinicalTrial, ChemblInteractions, CancerCommons
MAP2K1 5604 TAK-733 CHEMBL1615025 inhibitor MyCancerGenome, ClearityFoundationClinicalTrial, ChemblInteractions, CancerCommons
MAP2K1 5604 DABRAFENIB MESYLATE CHEMBL2105729 inhibitor MyCancerGenomeClinicalTrial
MAP2K1 5604 VEMURAFENIB CHEMBL1229517 CKB, CGI, CIViC, DoCM 21383288, 27312529, 24265153, 24448821, 22389471, 23569304, 7651428, 18632602, 25157968, 19915144, 22197931
MAP2K1 5604 DABRAFENIB CHEMBL2028663 CKB, CIViC 27312529, 24265153, 24265154, 22389471, 25370473, 24463458, 25673644
MAP2K1 5604 ENCORAFENIB CHEMBL3301612 CKB 27312529
MAP2K1 5604 OMIPALISIB CHEMBL1236962 CKB 22389471
MAP2K1 5604 BOSUTINIB CHEMBL288441 inhibitor DrugBank 19039322
MAP2K1 5604 TRAMETINIB CHEMBL2103875 inhibitor ClearityFoundationClinicalTrial, CGI, GuideToPharmacologyInteractions, OncoKB, TALC, CancerCommons, MyCancerGenome, MyCancerGenomeClinicalTrial, TdgClinicalTrial, CIViC, CKB 23846731, 25351745, 22663011, 26324360, 26566875, 25370473, 25673644, 27312529, 24265153, 28179366, 24265154, 26582713, 22389471, 26644315
MAP2K1 5604 CETUXIMAB CHEMBL1201577 CKB, CIViC 26644315, 27312529, 28179366
MAP2K1 5604 ALPELISIB CHEMBL2396661 CKB 27312529
MAP2K1 5604 RG-7167 CHEMBL3545383 inhibitor ChemblInteractions
MAP2K1 5604 AS-703988 CHEMBL3545243 inhibitor ChemblInteractions
MAP2K1 5604 TRAMETINIB DIMETHYL SULFOXIDE CHEMBL2105741 inhibitor ChemblInteractions
MAP2K1 5604 RG-7420 CHEMBL3330650 inhibitor ChemblInteractions
MAP2K1 5604 BALAMAPIMOD CHEMBL2104954 inhibitor ChemblInteractions
MAP2K1 5604 CHEMBL573819 CHEMBL573819 DrugBank 10592235
MAP2K1 5604 CHEMBL485945 CHEMBL485945 DrugBank 10592235
MAP2K1 5604 TOCILIZUMAB CHEMBL1237022 DrugBank 10592235
MAP2K1 5604 ARRY-300 CHEMBL3545359 TdgClinicalTrial
MAP2K1 5604 COBIMETINIB FUMARATE CHEMBL2364607 inhibitor ChemblInteractions
MAP2K1 5604 RG-7304 CHEMBL3545081 inhibitor ChemblInteractions
MAP2K1 5604 PD-0325901 CHEMBL507361 inhibitor TALC, MyCancerGenome, CKB, GuideToPharmacologyInteractions, ChemblInteractions, DrugBank, MyCancerGenomeClinicalTrial 26267534, 26582713, 10592235
MAP2K1 5604 BINIMETINIB CHEMBL3187723 inhibitor, allosteric modulator MyCancerGenome, TdgClinicalTrial, ClearityFoundationClinicalTrial, GuideToPharmacologyInteractions, ChemblInteractions, MyCancerGenomeClinicalTrial
MAP2K1 5604 SELUMETINIB CHEMBL1614701 inhibitor, allosteric modulator MyCancerGenome, CancerCommons, GuideToPharmacologyInteractions, TALC, ClearityFoundationClinicalTrial, MyCancerGenomeClinicalTrial, CIViC, CKB, ChemblInteractions 19915144, 26324360, 24448821, 22327936, 26582713, 22197931, 27312529, 25394791, 18632602
MAP2K1 5604 CHEMBL404939 CHEMBL404939 inhibitor GuideToPharmacologyInteractions
MAP2K1 5604 AZD-8330 CHEMBL3182621 inhibitor TALC, MyCancerGenome, TdgClinicalTrial, ChemblInteractions
MAP2K1 5604 WX-554 CHEMBL3545145 inhibitor TdgClinicalTrial, ChemblInteractions
MAP2K1 5604 Ro-4987655 CHEMBL1614766 inhibitor ChemblInteractions, CancerCommons
MAP2K1 5604 PANITUMUMAB CHEMBL1201827 CKB, CGI 26644315
MAP2K1 5604 CI-1040 CHEMBL105442 inhibitor, allosteric modulator MyCancerGenome, CKB, GuideToPharmacologyInteractions, ChemblInteractions 19915144, 12370306
MAP2K1 5604 Refametinib CHEMBL2138601 inhibitor, allosteric modulator GuideToPharmacologyInteractions, MyCancerGenomeClinicalTrial, CKB, MyCancerGenome, TALC, CancerCommons, ClearityFoundationClinicalTrial, ChemblInteractions 26582713
MAP2K1 5604 E-6201 CHEMBL1097999 inhibitor CKB, GuideToPharmacologyInteractions, ChemblInteractions 24448821
MAP2K1 5604 PLX-4720 CHEMBL1230020 CKB 21383288, 19915144
MAP2K1 5604 CERITINIB CHEMBL2403108 CKB 25394791

Variant-drug associations (data source: PharmGKB)
Gene Name Variant Alleles Chemical Phenotype Category Significance Notes Sentence Publications Annotation ID